SCHEMBL14977141

SCHEMBL14977141

O=C(O)C1CC(S(=O)(=O)c2ccccc2Cl)CN1C(=O)C1(c2ccc(Cl)cc2)CC1

nearest known ligand 0.73

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSL P07711 20/20 0.73
CTSB P07858 17/20 0.69
CTSS P25774 17/20 0.69
CTSK P43235 17/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3079583 1.00 CTSL (0.73) CTSLCTSBCTSSCTSK
SCHEMBL3067312 0.96 CTSL (0.68) CTSLCTSBCTSSCTSK
SCHEMBL3078477 0.95 CTSL (0.66) CTSLCTSBCTSSCTSK
SCHEMBL3076278 0.92 CTSL (0.73) CTSLCTSBCTSSCTSK
SCHEMBL14973560 0.92 CTSL (0.73) CTSLCTSBCTSSCTSK
SCHEMBL3060920 0.91 CTSL (0.62) CTSLCTSBCTSSCTSK
SCHEMBL3060809 0.90 CTSL (0.61) CTSLCTSBCTSSCTSK
SCHEMBL3071014 0.90 CTSL (0.61) CTSLCTSBCTSSCTSK
SCHEMBL3066405 0.90 CTSL (0.61) CTSLCTSBCTSSCTSK
SCHEMBL3064976 0.88 CTSL (0.65) CTSLCTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2782903-A1 NOVEL PYRROLIDINE DERIVATIVES AS INHIBITORS OF CATHEPSIN F.HOFFMANN-LA ROCHE AG (CH) 2014-10-01 EP disclosed
WO-2013076063-A1 NOVEL PYRROLIDINE DERIVATIVES AS INHIBITORS OF CATHEPSIN F. HOFFMANN-LA ROCHE AG (CH) 2013-05-30 WO disclosed