SCHEMBL14979102

SCHEMBL14979102

CNC(/C=C(\N)c1ccccc1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.43
TSHR P16473 3/20 0.43
CYP2C19 P33261 3/20 0.43
CYP2C9 P11712 2/20 0.43
PKM P14618 2/20 0.43
ADRA2C P18825 2/20 0.43
HSD17B10 Q99714 2/20 0.43
CHRM2 P08172 1/20 0.43
ADRA1A P35348 1/20 0.43
RGS12 O14924 1/20 0.43
GLA P06280 1/20 0.43
CYP2D6 P10635 1/20 0.43
ALOX15 P16050 1/20 0.43
ALOX12 P18054 1/20 0.43
NFKB1 P19838 1/20 0.43
HTR2A P28223 1/20 0.43
THPO P40225 1/20 0.43
GNAI1 P63096 1/20 0.43
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14979537 0.90 CYP3A4 (0.41) CYP3A4TSHRCYP2C19CYP2C9PKM
SCHEMBL14979110 0.79 CYP3A4 (0.43) CYP3A4TSHRCYP2C19CYP2C9PKM
SCHEMBL24534460 0.76 TRPA1 (0.52) CYP3A4TSHRCYP2C19CYP2C9PKM
SCHEMBL17449548 0.74
SCHEMBL21557737 0.74 CHRM2 (0.30) CYP3A4TSHRCYP2C19CYP2C9PKM
SCHEMBL11413560 0.73 DPP4 (0.41) CYP3A4TSHRCYP2C19PKMADRA2C
SCHEMBL16615163 0.73 DPP4 (0.41) CYP3A4TSHRCYP2C19PKMADRA2C
SCHEMBL8389881 0.72 BLM (0.41) CYP3A4TSHRCYP2C19PKMADRA2C
SCHEMBL21300718 0.71 EPHX2 (0.41) CYP3A4CYP2C19CYP2C9CYP2D6KMT2A
SCHEMBL18754634 0.71 BLM (0.39) CYP3A4TSHRCYP2C19PKMADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014038867-A1 A NOVEL COMBINATION OF A HOST COMPOUND AND A DOPANT COMPOUND AND AN ORGANIC ELECTROLUMINESCENCE DEVICE COMPRISING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2014-03-13 WO disclosed
WO-2013109045-A1 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2013-07-25 WO disclosed
WO-2013085243-A1 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2013-06-13 WO disclosed
WO-2013081416-A1 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2013-06-06 WO disclosed
WO-2013073874-A1 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUNDS AND AN ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2013-05-23 WO disclosed
WO-2013073896-A1 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2013-05-23 WO disclosed