SCHEMBL15033699

SCHEMBL15033699

CNc1ccc(N2CCC(C(F)(F)F)CC2)cc1C

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 1/20 0.36
MAPT P10636 4/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
HRH3 Q9Y5N1 9/20 0.35
KCNH2 Q12809 5/20 0.35
NOTUM Q6P988 1/20 0.34
RAD52 P43351 1/20 0.34
PDK2 Q15119 1/20 0.34
POLB P06746 1/20 0.34
CHRM3 P20309 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25042094 0.92 HRH3 (0.38) HRH3KCNH2NOTUMPDK2
SCHEMBL25042414 0.85 MAPT (0.40) ADRB1MAPTALDH1A1HRH3KCNH2
SCHEMBL9899784 0.84 S100B (0.36) MAPTKMT2AALDH1A1CYP1A2CYP2C9
SCHEMBL9939965 0.81 MAPT (0.36) MAPTKMT2AALDH1A1CYP1A2CYP2C9
SCHEMBL30279079 0.81 CHRM3 (0.39) MAPTALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL25039395 0.81 CHRM3 (0.39) MAPTALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL25042275 0.81 HRH4 (0.39) RAD52
SCHEMBL25187995 0.79 GAA (0.54) ADRB1MAPTKMT2AALDH1A1HPGD
SCHEMBL16727173 0.79 CCR1 (0.43) ADRB1MAPTALDH1A1NOTUM
SCHEMBL16181915 0.79 NR1H2 (0.36) MAPTKMT2AALDH1A1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8466186-B2 Compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-06-18 US disclosed