SCHEMBL15037486

SCHEMBL15037486

Cc1ccc(-c2ccc3nc(C)ccc3c2)cc1

nearest known ligand 0.70

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.70
KDM4E B2RXH2 1/20 0.55
LMNA P02545 1/20 0.55
POLB P06746 1/20 0.55
CASP6 P55212 1/20 0.55
BACE1 P56817 3/20 0.46
NCK1 P16333 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12923092 0.86 BACE1 (0.62) CYP1A2KDM4ELMNAPOLBCASP6
SCHEMBL982393 0.86 BACE1 (0.62) CYP1A2KDM4ELMNAPOLBCASP6
SCHEMBL16974223 0.85 CYP1A2 (0.55) CYP1A2KDM4ELMNAPOLBCASP6
SCHEMBL31307097 0.85 CYP1A2 (0.55) CYP1A2KDM4ELMNAPOLBCASP6
SCHEMBL29444268 0.83 CYP1A2 (1.00) CYP1A2KDM4ELMNAPOLBCASP6
SCHEMBL161703 0.83 CYP1A2 (1.00) CYP1A2KDM4ELMNAPOLBCASP6
SCHEMBL16574004 0.82 CYP1A2 (0.47) CYP1A2KDM4ELMNAPOLBCASP6
SCHEMBL12436949 0.82 CYP1A2 (0.52) CYP1A2KDM4ELMNAPOLBCASP6
Iodide SCHEMBL31142554 0.81 CYP1A2 (0.95) CYP1A2KDM4ELMNAPOLBCASP6
SCHEMBL28150727 0.81 BACE1 (0.54) CYP1A2KDM4ELMNABACE1NCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9127021-B2 Hepatitis C virus inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2015-09-08 US disclosed
US-8933110-B2 Hepatitis C virus inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2015-01-13 US disclosed
US-8785487-B2 Hepatitis C virus inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2014-07-22 US disclosed
WO-2013087743-A1 INHIBITORS OF HCV NS5A F. HOFFMANN-LA ROCHE AG (CH) 2013-06-20 WO disclosed