SCHEMBL15041527

SCHEMBL15041527

CC(C)n1c(=O)c(-c2ncc(S(=O)(=O)C3CCOCC3)cc2Cl)cc2cnc(Nc3ccc(OC4CCN(C)CC4)cc3)nc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 6/20 0.40
FGFR1 P11362 6/20 0.40
AXL P30530 5/20 0.40
PDGFRB P09619 3/20 0.40
PDGFRA P16234 3/20 0.40
SLC2A1 P11166 1/20 0.40
PKMYT1 Q99640 1/20 0.40
TNK2 Q07912 2/20 0.40
FGFR2 P21802 2/20 0.39
FGFR4 P22455 2/20 0.39
FGFR3 P22607 2/20 0.39
CCNB2 O95067 1/20 0.39
CCNE2 O96020 1/20 0.39
CDK1 P06493 1/20 0.39
CDK4 P11802 1/20 0.39
CCNB1 P14635 1/20 0.39
CCNA2 P20248 1/20 0.39
CCND1 P24385 1/20 0.39
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15041494 0.80 JAK2 (0.46) FGFR1AXLFGFR2FGFR4FGFR3
SCHEMBL15041499 0.74 CAMK2D (0.40) SRCFGFR1AXLPDGFRBTNK2
SCHEMBL15041896 0.73 TNK2 (0.39) SRCTNK2CAMK2DPAK4PKN1
SCHEMBL15041506 0.73 RIPK2 (0.42) SRCFGFR1AXLTNK2CAMK2D
SCHEMBL13553504 0.72 CAMK2D (0.40) SRCFGFR1AXLTNK2FGFR2
SCHEMBL15041887 0.72 FGFR1 (0.38) SRCFGFR1PDGFRBPDGFRAFGFR4
SCHEMBL15035114 0.72 PAK4 (0.40) SRCFGFR1AXLPDGFRBTNK2
SCHEMBL14682085 0.71 PKN1 (0.63) SRCFGFR1PDGFRBPDGFRASLC2A1
SCHEMBL15041858 0.71 TNK2 (0.41) SRCFGFR1TNK2CAMK2DPAK4
SCHEMBL15785236 0.71 PAK4 (0.43) SRCFGFR1AXLPDGFRBTNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8912203-B2 6-(sulfonylaryl)pyrido[2,3-D]pyrimidin-7(8H)-ones for the treatment of CNS disorders AFRAXIS HOLDINGS, INC. (US) 2014-12-16 US disclosed
US-20130158043-A1 PAK INHIBITORS FOR THE TREATMENT OF CANCER AFRAXIS, INC. (US) 2013-06-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130158043-A1 PAK INHIBITORS FOR THE TREATMENT OF CANCER PAK5, PAK2, PAK6 SRC 26/4885FGFR1 1919/4885AXL 1075/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.