SCHEMBL15054596

SCHEMBL15054596

CCOC(=O)C(=CNc1cccc(Br)c1F)C(=O)OCC

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.64
CYP2D6 P10635 2/20 0.64
DHODH Q02127 3/20 0.63
GAA P10253 3/20 0.63
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
NPSR1 Q6W5P4 5/20 0.52
MAPT P10636 6/20 0.50
KDM4E B2RXH2 5/20 0.50
LMNA P02545 3/20 0.50
MAPK1 P28482 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2C19 P33261 1/20 0.48
TDP1 Q9NUW8 1/20 0.46
ALDH1A1 P00352 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15054732 0.86 CYP3A4 (0.75) CYP3A4CYP2D6DHODHGAAMEN1
SCHEMBL17128366 0.86 DHODH (0.74) CYP3A4CYP2D6DHODHGAAMEN1
SCHEMBL31373277 0.84 CYP3A4 (0.64) CYP3A4CYP2D6DHODHGAAMEN1
SCHEMBL18987783 0.83 CYP3A4 (0.62) CYP3A4CYP2D6DHODHGAAMEN1
SCHEMBL11198142 0.83 DHODH (0.68) CYP3A4CYP2D6DHODHGAAMEN1
SCHEMBL2654418 0.82 CYP3A4 (0.61) CYP3A4CYP2D6DHODHGAAMEN1
SCHEMBL10862825 0.82 CYP3A4 (0.59) CYP3A4CYP2D6DHODHGAAMEN1
SCHEMBL25504852 0.82 MEN1 (0.60) CYP3A4CYP2D6DHODHGAAMEN1
SCHEMBL4154245 0.81 DHODH (0.74) CYP3A4CYP2D6DHODHGAAMEN1
SCHEMBL14845103 0.80 DHODH (0.64) CYP3A4CYP2D6DHODHGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013096151-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2013-06-27 WO disclosed