SCHEMBL2654418

SCHEMBL2654418

CCOC(=O)C(=CNc1cccc(C(F)(F)F)c1F)C(=O)OCC

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.61
CYP2D6 P10635 2/20 0.61
DHODH Q02127 3/20 0.60
GAA P10253 2/20 0.60
NPSR1 Q6W5P4 5/20 0.60
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
KDM4E B2RXH2 5/20 0.51
LMNA P02545 2/20 0.51
MAPK1 P28482 2/20 0.51
POLB P06746 1/20 0.48
MAPT P10636 4/20 0.48
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
EPHX2 P34913 1/20 0.46
TDP1 Q9NUW8 1/20 0.44
CTSS P25774 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1124285 0.88 DHODH (0.68) CYP3A4CYP2D6DHODHGAANPSR1
SCHEMBL11403188 0.82 DHODH (0.60) CYP3A4CYP2D6DHODHGAANPSR1
SCHEMBL15054596 0.82 CYP3A4 (0.64) CYP3A4CYP2D6DHODHGAANPSR1
SCHEMBL18987783 0.81 CYP3A4 (0.62) CYP3A4CYP2D6DHODHGAANPSR1
SCHEMBL995708 0.80 DHODH (0.56) CYP3A4CYP2D6DHODHGAANPSR1
SCHEMBL995706 0.80 DHODH (0.56) CYP3A4CYP2D6DHODHGAANPSR1
SCHEMBL4154245 0.79 DHODH (0.74) CYP3A4CYP2D6DHODHGAANPSR1
SCHEMBL2654421 0.78 EPHX2 (0.42) CYP3A4CYP2D6DHODHGAANPSR1
SCHEMBL8628152 0.78 DHODH (0.59) CYP3A4CYP2D6DHODHGAANPSR1
SCHEMBL31373277 0.77 CYP3A4 (0.64) CYP3A4CYP2D6DHODHGAANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004043930-A1 QUINOLINE DERIVATIVES WHICH ENHANCE COGNITION VIA THE GABA-A RECEPTOR MERCK SHARP & DOHME LIMITED (GB) 2004-05-27 WO disclosed