SCHEMBL1505907

SCHEMBL1505907

Fc1ccc([C@H]2CO2)cc1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.56
KDM1A O60341 2/20 0.44
SLC6A2 P23975 2/20 0.43
HTR2A P28223 2/20 0.43
HTR2C P28335 2/20 0.43
SLC6A4 P31645 2/20 0.43
HTR2B P41595 2/20 0.43
SLC6A3 Q01959 2/20 0.43
MAOB P27338 5/20 0.42
ATM Q13315 1/20 0.41
FADS1 O60427 2/20 0.41
CYP19A1 P11511 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL937356 1.00 TSHR (0.56) TSHRKDM1ASLC6A2HTR2AHTR2C
SCHEMBL1505987 1.00 TSHR (0.56) TSHRKDM1ASLC6A2HTR2AHTR2C
SCHEMBL46155 0.86 TSHR (0.72) TSHR
SCHEMBL16422345 0.81 KDM1A (0.48) TSHRKDM1ASLC6A2HTR2AHTR2C
SCHEMBL21353917 0.81 KDM1A (0.39) TSHRKDM1ASLC6A2HTR2AHTR2C
SCHEMBL21363715 0.81 KDM1A (0.39) TSHRKDM1ASLC6A2HTR2AHTR2C
SCHEMBL21353919 0.81 KDM1A (0.39) TSHRKDM1ASLC6A2HTR2AHTR2C
SCHEMBL21393372 0.81 KDM1A (0.39) TSHRKDM1ASLC6A2HTR2AHTR2C
SCHEMBL16423075 0.81 KDM1A (0.48) TSHRKDM1ASLC6A2HTR2AHTR2C
SCHEMBL16422344 0.81 KDM1A (0.48) TSHRKDM1ASLC6A2HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 78 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11773068-B2 KDM1A inhibitors for the treatment of disease IMAGO BIOSCIENCES, INC. (US) 2023-10-03 US disclosed
US-11773068-B2 KDM1A inhibitors for the treatment of disease IMAGO BIOSCIENCES, INC. (US) 2023-10-03 US disclosed
US-11655226-B2 KDM1A inhibitors for the treatment of disease IMAGO BIOSCIENCES, INC. (US) 2023-05-23 US disclosed
US-11655226-B2 KDM1A inhibitors for the treatment of disease IMAGO BIOSCIENCES, INC. (US) 2023-05-23 US disclosed
US-20230000835-A1 LYSINE-SPECIFIC HISTONE DEMETHYLASE INHIBITORS FOR THE TREATMENT OF MYELOPROLIFERATIVE NEOPLASMS IMAGO BIOSCIENCES, INC. 2023-01-05 US disclosed
US-20220025424-A1 COMPOSITIONS AND METHODS FOR PRODUCING STEREOISOMERICALLY PURE AMINOCYCLOPROPANES IMAGO BIOSCIENCES, INC. 2022-01-27 US disclosed
US-20220025424-A1 COMPOSITIONS AND METHODS FOR PRODUCING STEREOISOMERICALLY PURE AMINOCYCLOPROPANES IMAGO BIOSCIENCES, INC. 2022-01-27 US disclosed
US-11230534-B2 KDM1A inhibitors for the treatment of disease IMAGO BIOSCIENCES, INC. (US) 2022-01-25 US disclosed
US-20210386733-A1 LYSINE-SPECIFIC HISTONE DEMETHYLASE INHIBITORS FOR THE TREATMENT OF MYELOPROLIFERATIVE NEOPLASMS IMAGO BIOSCIENCES, INC. 2021-12-16 US disclosed
US-20210196711-A1 LYSINE-SPECIFIC HISTONE DEMETHYLASE AS A NOVEL THERAPEUTIC TARGET IN MYELOPROLIFERATIVE NEOPLASMS IMAGO BIOSCIENCES, INC. 2021-07-01 US disclosed
WO-2008064817-A2 METHOD FOR THE STEREOSELECTIVE SYNTHESIS OF CHIRAL EPOXIDES BY ADH REDUCTION OF KETONES SUBSTITUTED WITH ALPHA STARTING GROUPS AND CYCLISATION ARCHIMICA GMBH (DE) 2008-06-05 WO disclosed
EP-1910320-A2 INTERMEDIATE COMPOUND FOR SYNTHESIZING PHARMACEUTICAL AGENT AND PRODUCTION METHOD THEREOF Mitsubishi Tanabe Pharma Corporation (JP) 2008-04-16 EP disclosed
EP-1899313-A1 METHOD FOR PRODUCING SINGLE ENANTIOMER EPOXIDES BY THE ADH REDUCTION OF ALPHA-LEAVING GROUP-SUBSTITUTED KETONES AND CYCLISATION Archimica GmbH (DE) 2008-03-19 EP disclosed
WO-2007113309-A2 COMPOUNDS WHICH INHIBIT THE GLYCINE TRANSPORTER AND USES THEREOF GLAXO GROUP LIMITED (GB) 2007-10-11 WO disclosed
WO-2007011065-A2 INTERMEDIATE COMPOUND FOR SYNTHESIZING PHARMACEUTICAL AGENT AND PRODUCTION METHOD THEREOF MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-01-25 WO disclosed
EP-1742921-A2 PYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF CANCER AstraZeneca AB (SE) 2007-01-17 EP disclosed
WO-2006136289-A1 METHOD FOR PRODUCING SINGLE ENANTIOMER EPOXIDES BY THE ADH REDUCTION OF ALPHA-LEAVING GROUP-SUBSTITUTED KETONES AND CYCLISATION ARCHIMICA GMBH (DE) 2006-12-28 WO disclosed
WO-2005103010-A2 PYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF CANCER ASTRAZENECA AB (SE) 2005-11-03 WO disclosed
EP-1043319-B1 NOVEL ALKYLAMINO DERIVATIVES MITSUBISHI CHEM CORP (JP) 2005-03-16 EP disclosed
EP-1043319-A1 NOVEL ALKYLAMINO DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2000-10-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210386733-A1 LYSINE-SPECIFIC HISTONE DEMETHYLASE INHIBITORS FOR THE TREATMENT OF MYELOPROLIFERATIVE NEOPLASMS KDM1B, KDM1A, KDM3A TSHR 3821/4885KDM1A 2/4885SLC6A2 4083/4885
US-20210196711-A1 LYSINE-SPECIFIC HISTONE DEMETHYLASE AS A NOVEL THERAPEUTIC TARGET IN MYELOPROLIFERATIVE NEOPLASMS KDM1B, KDM1A, KDM2A TSHR 3736/4885KDM1A 2/4885SLC6A2 3976/4885
US-11230534-B2 KDM1A inhibitors for the treatment of disease KDM1B, KDM1A, KDM2A TSHR 4247/4885KDM1A 2/4885SLC6A2 4581/4885
US-20230000835-A1 LYSINE-SPECIFIC HISTONE DEMETHYLASE INHIBITORS FOR THE TREATMENT OF MYELOPROLIFERATIVE NEOPLASMS KDM1B, KDM1A, KDM3A TSHR 3821/4885KDM1A 2/4885SLC6A2 4083/4885
US-11773068-B2 KDM1A inhibitors for the treatment of disease KDM1B, KDM1A, KDM2A TSHR 4247/4885KDM1A 2/4885SLC6A2 4581/4885
US-11655226-B2 KDM1A inhibitors for the treatment of disease KDM1B, KDM1A, KDM2A TSHR 4247/4885KDM1A 2/4885SLC6A2 4581/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.