SCHEMBL15060022

SCHEMBL15060022

Cn1cc(Nc2ncc(Cl)c(NC[C@@H]3CCNC3)n2)cn1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 9/20 0.58
JAK2 O60674 8/20 0.58
CDK19 Q9BWU1 1/20 0.54
ALK Q9UM73 1/20 0.54
JAK3 P52333 3/20 0.52
TYK2 P29597 2/20 0.52
AURKB Q96GD4 6/20 0.51
KDR P35968 5/20 0.51
AURKA O14965 6/20 0.50
CDC7 O00311 1/20 0.48
DAPK3 O43293 1/20 0.48
ROCK2 O75116 1/20 0.48
PRKD3 O94806 1/20 0.48
MAP4K4 O95819 1/20 0.48
PAK4 O96013 1/20 0.48
PIM1 P11309 1/20 0.48
PRKACA P17612 1/20 0.48
CDK2 P24941 1/20 0.48
SYK P43405 1/20 0.48
CSNK1A1 P48729 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL15059314 0.99 JAK1 (0.57) JAK1JAK2CDK19ALKJAK3
SCHEMBL16336889 0.94 JAK1 (0.56) JAK1JAK2CDK19ALKJAK3
SCHEMBL15059571 0.94 JAK1 (0.56) JAK1JAK2CDK19ALKJAK3
SCHEMBL16337387 0.94 JAK1 (0.56) JAK1JAK2CDK19ALKJAK3
SCHEMBL16336520 0.89 JAK1 (0.52) JAK1JAK2JAK3TYK2AURKB
SCHEMBL15059525 0.88 JAK2 (0.55) JAK1JAK2JAK3TYK2AURKB
SCHEMBL15059526 0.88 JAK2 (0.55) JAK1JAK2JAK3TYK2AURKB
SCHEMBL16337487 0.88 JAK2 (0.55) JAK1JAK2JAK3TYK2AURKB
SCHEMBL15059873 0.85 CDK19 (0.58) JAK1JAK2CDK19ALKJAK3
SCHEMBL15071983 0.83 JAK2 (0.58) JAK1JAK2CDK19ALKJAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2794598-A1 PYRIMIDINE-2,4-DIAMINE DERIVATIVES AS KINASE INHIBITORS Cellzome Limited (GB) 2014-10-29 EP disclosed
WO-2013092854-A1 PYRIMIDINE-2,4-DIAMINE DERIVATIVES AS KINASE INHIBITORS CELLZOME LIMITED (GB) 2013-06-27 WO disclosed