SCHEMBL15062004

SCHEMBL15062004

Cc1ccccc1OC1CCN(C)C1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.51
SCD O00767 1/20 0.49
HTR2C P28335 3/20 0.48
HTR2B P41595 3/20 0.48
NOS3 P29474 1/20 0.47
NOS1 P29475 1/20 0.47
NOS2 P35228 1/20 0.47
CHRM4 P08173 1/20 0.47
CHRM5 P08912 1/20 0.47
CHRM1 P11229 1/20 0.47
CHRM3 P20309 1/20 0.47
EPHX2 P34913 1/20 0.45
HRH1 P35367 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10260949 1.00 PDE10A (0.51) PDE10ASCDHTR2CHTR2BNOS3
SCHEMBL10260935 1.00 PDE10A (0.51) PDE10ASCDHTR2CHTR2BNOS3
SCHEMBL10274501 0.91 SCD (0.53) PDE10ASCDCHRM4CHRM5CHRM1
SCHEMBL30656257 0.91 SCD (0.53) PDE10ASCDCHRM4CHRM5CHRM1
SCHEMBL10260948 0.87 SLC6A4 (0.44) PDE10ASCDCHRM4CHRM3
SCHEMBL14578204 0.84 HTR2C (0.53) HTR2CHTR2BNOS3NOS1NOS2
SCHEMBL10261314 0.81 HTR2C (0.51) HTR2CHTR2BNOS3NOS1NOS2
SCHEMBL1927488 0.81 UTS2R (0.51) HTR2CHTR2BNOS3NOS1NOS2
SCHEMBL15651062 0.81 NOS3 (0.52) HTR2CHTR2BNOS3NOS1NOS2
SCHEMBL10260926 0.81 HTR2C (0.51) HTR2CHTR2BNOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2607364-A1 Tetraaza-cyclopenta[a]indenyl and their use as positive allosteric modulators Ares Trading S.A. (CH) 2013-06-26 EP disclosed