SCHEMBL15069746

SCHEMBL15069746

COc1ccc(Nc2nccc3c(Nc4ccsc4)c(C)ccc23)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIP4K2A P48426 9/20 0.44
BRAF P15056 3/20 0.42
CSF1R P07333 2/20 0.42
RAF1 P04049 1/20 0.42
DDR1 Q08345 1/20 0.42
DDR2 Q16832 1/20 0.42
MAPT P10636 3/20 0.41
GRM4 Q14833 1/20 0.41
LMNA P02545 2/20 0.41
TP53 P04637 1/20 0.41
LCK P06239 2/20 0.41
TEK Q02763 2/20 0.41
KDR P35968 1/20 0.41
TNF P01375 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
POLB P06746 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15069754 0.86 BRAF (0.55) BRAFCSF1RRAF1DDR1DDR2
SCHEMBL15069728 0.86 BRAF (0.42) BRAFCSF1RRAF1DDR1DDR2
SCHEMBL15068707 0.83 BRAF (0.55) BRAFCSF1RRAF1DDR1DDR2
SCHEMBL15069738 0.82 BRAF (0.45) BRAFCSF1RRAF1DDR1DDR2
SCHEMBL15069205 0.81 BRAF (0.44) BRAFCSF1RRAF1DDR1DDR2
SCHEMBL15066146 0.81 PIK3CG (0.41) PIP4K2ABRAFCSF1RRAF1DDR1
SCHEMBL15069808 0.81 BRAF (0.43) BRAFCSF1RRAF1DDR1DDR2
SCHEMBL26373434 0.79 PIP4K2A (0.50) PIP4K2AMAPTGRM4LMNATP53
SCHEMBL15069790 0.79 BRAF (0.43) BRAFCSF1RRAF1DDR1DDR2
SCHEMBL15069219 0.79 BRAF (0.44) BRAFCSF1RRAF1DDR1DDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2797927-A1 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY FOR PROTEIN KINASES Hanmi Pharm. Co., Ltd. (KR) 2014-11-05 EP disclosed
WO-2013100632-A1 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY FOR PROTEIN KINASES HANMI PHARM CO., LTD. (KR) 2013-07-04 WO disclosed