SCHEMBL1507316

SCHEMBL1507316

O=C(NCC1OCCO1)c1cc(C(=O)c2c(F)cc(F)cc2F)c[nH]1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.48
HPGD P15428 4/20 0.47
ALDH1A1 P00352 4/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C19 P33261 1/20 0.47
MAPK14 Q16539 6/20 0.47
MAPK7 Q13164 2/20 0.47
HTT P42858 3/20 0.46
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10042102 0.80 MAPK14 (0.52) L3MBTL1MAPK14MAPK7HTT
SCHEMBL299630 0.72 POLB (0.50) ALDH1A1MAPK14MAPK7LMNA
SCHEMBL297517 0.71 MAPK14 (0.47) ALDH1A1MAPK14MAPK7HTTLMNA
SCHEMBL10042100 0.70 POLB (0.49) ALDH1A1MAPK14MAPK7HTTLMNA
SCHEMBL298823 0.70 MAPK14 (0.46) ALDH1A1CYP1A2CYP2C19MAPK14MAPK7
SCHEMBL606462 0.70 MAPK14 (0.46) ALDH1A1CYP1A2CYP2C19MAPK14MAPK7
SCHEMBL298824 0.70 BAZ2B (0.55) ALDH1A1MAPK14MAPK7HTTLMNA
SCHEMBL10042044 0.70 MAPK14 (0.50) L3MBTL1HPGDALDH1A1CYP1A2CYP2C19
SCHEMBL13074869 0.69 MAPK14 (0.44) L3MBTL1MAPK14MAPK7HTT
SCHEMBL13074868 0.68 HTT (0.49) HPGDALDH1A1CYP1A2CYP2C19MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2300485-A1 PYRROLO Ý2, 3-C¨PYRIDINE DERIVATIVES AS P38 KINASE INHIBITING AGENTS Merck Sharp & Dohme Corp. (US) 2011-03-30 EP disclosed