SCHEMBL15073265

SCHEMBL15073265

O=C(O)C[C@H]1CC[C@H](c2ccc(-c3ccc(-c4nnc(-c5ccccc5)[nH]4)cc3)cc2)CC1

nearest known ligand 0.58

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 19/20 0.58
SOAT1 P35610 3/20 0.58
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15073180 0.89 DGAT1 (0.62) DGAT1SOAT1
SCHEMBL3538810 0.79 IDO1 (0.57) DGAT1SOAT1NPC1RAB9A
SCHEMBL17318281 0.79 IDO1 (0.57) DGAT1SOAT1NPC1RAB9A
SCHEMBL3538808 0.79 IDO1 (0.57) DGAT1SOAT1NPC1RAB9A
SCHEMBL4940938 0.78 DGAT1 (0.59) DGAT1SOAT1
SCHEMBL4939294 0.77 DGAT1 (0.53) DGAT1SOAT1
SCHEMBL902399 0.76 DGAT1 (0.60) DGAT1SOAT1
SCHEMBL15073300 0.76 ESR2 (0.42) DGAT1SOAT1NPC1RAB9A
SCHEMBL902462 0.75 DGAT1 (0.73) DGAT1SOAT1
SCHEMBL16649074 0.74 DGAT1 (0.60) DGAT1SOAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013096093-A1 COMPOUNDS AS DGAT-1 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-06-27 WO disclosed