SCHEMBL1507426

SCHEMBL1507426

O=C(O)c1cc(C(=O)c2cccc(F)c2F)c[nH]1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 9/20 0.59
MAPK7 Q13164 3/20 0.59
POLB P06746 2/20 0.51
ALDH1A1 P00352 3/20 0.47
PKM P14618 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
RAB9A P51151 2/20 0.47
NPC1 O15118 1/20 0.47
HSP90AA1 P07900 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CES2 O00748 1/20 0.46
BCHE P06276 1/20 0.46
CES1 P23141 1/20 0.46
MTNR1A P48039 1/20 0.46
MTNR1B P49286 1/20 0.46
GAA P10253 1/20 0.46
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17607058 0.88 MAPK14 (0.67) MAPK14MAPK7POLBALDH1A1PKM
SCHEMBL300049 0.84 POLB (0.68) MAPK14MAPK7POLBALDH1A1PKM
SCHEMBL29191087 0.83 MAPK14 (0.57) MAPK14MAPK7POLBALDH1A1GAA
SCHEMBL17607070 0.78 MAPK7 (0.63) MAPK14MAPK7POLBALDH1A1PKM
SCHEMBL17607056 0.78 POLB (0.60) MAPK14MAPK7POLBALDH1A1PKM
SCHEMBL31114409 0.78 MAPK7 (0.63) MAPK14MAPK7POLBALDH1A1PKM
SCHEMBL298049 0.78 KMT2A (0.71) MAPK14POLBALDH1A1PKML3MBTL1
SCHEMBL10756348 0.77 CDC25B (0.55) MAPK14POLBALDH1A1PKML3MBTL1
SCHEMBL4827330 0.76 RAB9A (0.59) MAPK14MAPK7POLBALDH1A1PKM
SCHEMBL5038336 0.76 GAA (0.49) MAPK14MAPK7ALDH1A1RAB9ACES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117886734-A Heterocyclic amide compound and preparation method, pharmaceutical composition and application thereof 中国药科大学 2024-04-16 CN disclosed
EP-2300485-A1 PYRROLO Ý2, 3-C¨PYRIDINE DERIVATIVES AS P38 KINASE INHIBITING AGENTS Merck Sharp & Dohme Corp. (US) 2011-03-30 EP disclosed
WO-2009152072-A1 PYRROLO [2, 3-C] PYRIDINE DERIVATIVES AS P38 KINASE INHIBITING AGENTS MERCK & CO., INC. (US) 2009-12-17 WO disclosed