Fluorescin

Fluorescin

SCHEMBL1507667

O=C(O)c1ccccc1C1c2ccc(O)cc2Oc2cc(O)ccc21.[KH]

nearest known ligand 0.69

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.69
ALDH1A1 P00352 4/20 0.52
HSD17B10 Q99714 3/20 0.52
BRCA1 P38398 2/20 0.52
CYP3A4 P08684 1/20 0.52
HPGD P15428 1/20 0.52
ALOX15 P16050 1/20 0.52
ALOX12 P18054 1/20 0.52
CASP1 P29466 1/20 0.52
STAT6 P42226 1/20 0.52
CASP7 P55210 1/20 0.52
HBB P68871 1/20 0.52
HIF1A Q16665 1/20 0.52
ESR1 P03372 5/20 0.48
ESR2 Q92731 3/20 0.48
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
USP2 O75604 2/20 0.46
POLB P06746 1/20 0.46
HSP90AA1 P07900 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fluorescin SCHEMBL31164674 0.98 CYP2C9 (0.71) CYP2C9ALDH1A1HSD17B10BRCA1CYP3A4
Fluorescin SCHEMBL31164673 0.98 CYP2C9 (0.71) CYP2C9ALDH1A1HSD17B10BRCA1CYP3A4
Fluorescin SCHEMBL29370997 0.98 CYP2C9 (0.71) CYP2C9ALDH1A1HSD17B10BRCA1CYP3A4
Fluorescin SCHEMBL31214151 0.98 CYP2C9 (0.71) CYP2C9ALDH1A1HSD17B10BRCA1CYP3A4
Fluorescin SCHEMBL27403 0.98 CYP2C9 (0.71) CYP2C9ALDH1A1HSD17B10BRCA1CYP3A4
Fluorescin SCHEMBL1938032 0.97 CYP2C9 (0.69) CYP2C9ALDH1A1HSD17B10BRCA1CYP3A4
Fluorescin SCHEMBL5579981 0.93 CYP2C9 (0.64) CYP2C9ALDH1A1HSD17B10BRCA1CYP3A4
Fluorescin SCHEMBL7807189 0.93 CYP2C9 (0.64) CYP2C9ALDH1A1HSD17B10BRCA1CYP3A4
Fluorescin SCHEMBL4342272 0.93 CYP2C9 (0.64) CYP2C9ALDH1A1HSD17B10BRCA1CYP3A4
Fluorescin SCHEMBL6036317 0.92 CYP2C9 (0.62) CYP2C9ALDH1A1HSD17B10BRCA1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2305246-B1 Tumor necrosis factor inhibitors UNIV PENNSYLVANIA (US) 2015-08-26 EP disclosed
US-9096607-B2 Tumor necrosis factor inhibitors THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2015-08-04 US disclosed
US-20140256803-A1 TUMOR NECROSIS FACTOR INHIBITORS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2014-09-11 US disclosed
US-8765810-B2 Tumor necrosis factor inhibitors THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2014-07-01 US disclosed
EP-2298295-B1 Tumor necrosis factor inhibitors CEPHALON INC (US) 2013-08-28 EP disclosed
US-20130072562-A1 TUMOR NECROSIS FACTOR INHIBITORS CEPHALON, INC. (US) 2013-03-21 US disclosed
US-8318699-B2 Tumor necrosis factor inhibitors THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2012-11-27 US disclosed
EP-2305246-A1 Tumor necrosis factor inhibitors Ception Therapeutics, Inc. (US) 2011-04-06 EP disclosed
EP-2298295-A1 Tumor necrosis factor inhibitors Ception Therapeutics, Inc. (US) 2011-03-23 EP disclosed
US-20090221527-A1 TUMOR NECROSIS FACTOR INHIBITORS CEPTION THERAPEUTICS, INC. (US) 2009-09-03 US disclosed
EP-1845970-A4 TUMOR NECROSIS FACTOR INHIBITORS CEPTION THERAPEUTICS INC (US) 2009-02-18 EP disclosed
EP-1845970-A2 TUMOR NECROSIS FACTOR INHIBITORS Ception Therapeutics, Inc. (US) 2007-10-24 EP disclosed
WO-2006083970-A2 TUMOR NECROSIS FACTOR INHIBITORS CEPTION THERAPEUTICS, INC. (US) 2006-08-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090221527-A1 TUMOR NECROSIS FACTOR INHIBITORS TNFRSF1A, TNF, TNFRSF9 CYP2C9 4775/4885ALDH1A1 3912/4885HSD17B10 3180/4885
US-20140256803-A1 TUMOR NECROSIS FACTOR INHIBITORS TNFRSF1A, TNF, TNFRSF9 CYP2C9 4775/4885ALDH1A1 3912/4885HSD17B10 3180/4885
US-20130072562-A1 TUMOR NECROSIS FACTOR INHIBITORS TNFRSF1A, TNF, TNFRSF9 CYP2C9 4775/4885ALDH1A1 3912/4885HSD17B10 3180/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.