SCHEMBL15076909

SCHEMBL15076909

CC(=O)Nc1cc(-c2cc(-c3nnc[nH]3)c[nH]2)ccn1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIK3C3 Q8NEB9 18/20 0.47
GSK3B P49841 1/20 0.41
MAPK14 Q16539 1/20 0.41
PIP5K1C O60331 1/20 0.40
PIK3CA P42336 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28124623 0.78 PIK3C3 (0.51) PIK3C3PIP5K1CPIK3CA
SCHEMBL15051235 0.76 PIK3C3 (0.43) PIK3C3GSK3BMAPK14
SCHEMBL15051156 0.76 PIK3C3 (0.42) PIK3C3GSK3BMAPK14PIP5K1CPIK3CA
SCHEMBL15050809 0.72 PIK3C3 (0.52) PIK3C3MAPK14
SCHEMBL19736124 0.72 PIK3C3 (0.57) PIK3C3
SCHEMBL953124 0.71 MAPK14 (0.47) PIK3C3MAPK14PIP5K1CPIK3CA
SCHEMBL953912 0.71 MAPK14 (0.42) PIK3C3GSK3BMAPK14
SCHEMBL12852676 0.70 ROCK2 (0.41) PIK3C3MAPK14
SCHEMBL19706510 0.70 PIK3C3 (0.62) PIK3C3
SCHEMBL16850488 0.69 GSK3B (0.44) PIK3C3GSK3BMAPK14PIP5K1CPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013096637-A1 HETEROARYLS AND USES THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2013-06-27 WO disclosed