SCHEMBL15077170

SCHEMBL15077170

CN(C)Cc1cc(C(C)(C)C)cc(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
GAA P10253 1/20 0.47
TSHR P16473 1/20 0.47
TACR1 P25103 10/20 0.44
CYP1A2 P05177 1/20 0.42
IDO1 P14902 2/20 0.41
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
LSS P48449 1/20 0.39
CETP P11597 1/20 0.38
SERPINE1 P05121 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13451382 0.92 TACR1 (0.49) ALDH1A1LMNAGAATSHRTACR1
SCHEMBL14007668 0.90 CYP2C19 (0.55) CYP2C19ALDH1A1LMNAGAATSHR
SCHEMBL15077173 0.81 TACR1 (0.46) TACR1IDO1
SCHEMBL15078647 0.81 TACR1 (0.41) ALDH1A1LMNAGAATSHRTACR1
SCHEMBL10104524 0.81 TACR1 (0.41) ALDH1A1LMNAGAATSHRTACR1
SCHEMBL13178016 0.79 TACR1 (0.61) TACR1IDO1SERPINE1
SCHEMBL788092 0.79 TACR1 (0.40) ALDH1A1LMNAGAATSHRTACR1
SCHEMBL12305670 0.79 ALDH1A1 (0.46) CYP2C19ALDH1A1LMNAGAATSHR
SCHEMBL30950869 0.79 TACR1 (0.40) ALDH1A1LMNAGAATSHRTACR1
SCHEMBL345830 0.79 SLC6A4 (0.43) ALDH1A1LMNAGAATSHRTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130165440-A1 JAK1 Inhibitors EXELIXIS, INC. (US) 2013-06-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130165440-A1 JAK1 Inhibitors JAK1, JAK2, JAK3 CYP2C19 1695/4885ALDH1A1 1886/4885LMNA 4206/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.