SCHEMBL1507873

SCHEMBL1507873

N#Cc1ccc(Cn2ccnc2Cc2ccccc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 5/20 0.48
CYP11B2 P19099 5/20 0.48
HSP90AA1 P07900 2/20 0.47
HSP90B1 P14625 1/20 0.46
CYP19A1 P11511 6/20 0.45
KMT2A Q03164 2/20 0.44
MMP13 P45452 1/20 0.43
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
ALOX12 P18054 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30610947 1.00 CYP11B1 (0.48) CYP11B1CYP11B2HSP90AA1HSP90B1CYP19A1
Hydrochloric Acid SCHEMBL1507947 0.99 CYP11B1 (0.47) CYP11B1CYP11B2HSP90AA1HSP90B1CYP19A1
SCHEMBL1508003 0.94 CYP19A1 (0.50) CYP11B1CYP11B2HSP90AA1HSP90B1CYP19A1
SCHEMBL1508007 0.88 HSP90AA1 (0.50) CYP11B1CYP11B2HSP90AA1HSP90B1CYP19A1
SCHEMBL1723554 0.87 HSP90AA1 (0.57) CYP11B1CYP11B2HSP90AA1HSP90B1KMT2A
Hydrochloric Acid SCHEMBL4053167 0.85 HSP90AA1 (0.56) HSP90AA1HSP90B1KMT2AMEN1ALDH1A1
SCHEMBL6981310 0.84 HSP90AA1 (0.42) CYP11B1CYP11B2HSP90AA1HSP90B1CYP19A1
SCHEMBL4978567 0.83 HSP90AA1 (0.41) CYP11B1CYP11B2HSP90AA1HSP90B1KMT2A
SCHEMBL3403218 0.81 SMN1; SMN2 (0.52) CYP11B1CYP11B2HSP90AA1HSP90B1KMT2A
SCHEMBL3338535 0.81 HSP90AA1 (0.50) HSP90AA1HSP90B1KMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0236940-B3 Alpha-heterocycle substituted tolunitriles NOVARTIS AG (CH) 2011-03-23 EP claimed
EP-0236940-B1 ALPHA-HETEROCYCLE SUBSTITUTED TOLUNITRILES CIBA-GEIGY AG (CH) 1993-09-22 EP claimed
EP-0236940-A2 Alpha-heterocycle substituted tolunitriles CIBA-GEIGY AG (CH) 1987-09-16 EP claimed