Oxalic Acid

Oxalic Acid

SCHEMBL1507978

CCCCC(c1ccc(C#N)cc1)c1ncc[nH]1.O=C(O)C(=O)O

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1SLC6A4

The experimentally established mechanism targets of Oxalic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA2C P18825 1/20 0.42
CYP19A1 P11511 8/20 0.41
PTGES O14684 1/20 0.38
ALOX5 P09917 1/20 0.38
PPARG P37231 1/20 0.38
FPR2 P25090 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
KDM4E B2RXH2 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MGLL Q99685 1/20 0.35
EPHX2 P34913 1/20 0.35
MMP2 P08253 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10686017 0.94 CYP19A1 (0.45) CYP19A1PTGESALOX5PPARGCYP1A2
SCHEMBL11223097 0.79 SLC6A4 (0.45) ADRA2AADRA2BCYP19A1CYP3A4CYP2D6
SCHEMBL9803992 0.79 CYP19A1 (0.43) ADRA2AADRA2BADRA2CCYP19A1FPR2
SCHEMBL7908696 0.77 CYP19A1 (0.42) ADRA2AADRA2BADRA2CCYP19A1FPR2
SCHEMBL8411281 0.76 CYP19A1 (0.63) CYP19A1EPHX2SLC6A3
SCHEMBL8326961 0.76 CYP19A1 (0.37) ADRA2AADRA2BADRA2CCYP19A1CYP2C9
SCHEMBL19642925 0.75 CYP1A2 (0.44) ADRA2AADRA2BADRA2CCYP19A1FPR2
SCHEMBL30585956 0.75 CYP19A1 (0.51) CYP19A1KDM4EGAAMAPTL3MBTL1
SCHEMBL6437501 0.75 CYP19A1 (0.41) CYP19A1
Succinic Acid SCHEMBL1649163 0.74 MMP2 (0.42) ADRA2AADRA2BADRA2CCYP19A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0236940-B3 Alpha-heterocycle substituted tolunitriles NOVARTIS AG (CH) 2011-03-23 EP disclosed
US-5473078-A Aromatase inhibiting compounds CIBA-GEIGY CORPORATION (US) 1995-12-05 US disclosed
US-5352795-A Condensing triazolylmethylbenzonitrile with fluorobenzonitrile under basic conditions using alkali metal alkoxide CIBA-GEIGY CORPORATION (US) 1994-10-04 US disclosed
EP-0236940-B1 ALPHA-HETEROCYCLE SUBSTITUTED TOLUNITRILES CIBA-GEIGY AG (CH) 1993-09-22 EP disclosed
US-5112845-A Inhibitors of estrogen synthesis, veterinary medicine CIBA-GEIGY CORPORATION (US) 1992-05-12 US disclosed
US-4978672-A Alpha-heterocyclc substituted tolunitriles CIBA-GEIGY CORPORATION (US) 1990-12-18 US disclosed
EP-0236940-A2 Alpha-heterocycle substituted tolunitriles CIBA-GEIGY AG (CH) 1987-09-16 EP disclosed