SCHEMBL15084518

SCHEMBL15084518

COc1cc2ncnc(Oc3ccc(N)cc3F)c2cc1OCCCN1CCN(C)CC1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.67
FLT4 P35916 7/20 0.67
AURKB Q96GD4 4/20 0.67
PDGFRB P09619 3/20 0.67
TEK Q02763 3/20 0.67
AURKA O14965 3/20 0.67
AXL P30530 6/20 0.65
EGFR P00533 7/20 0.58
FLT1 P17948 5/20 0.58
FGFR1 P11362 4/20 0.58
RET P07949 3/20 0.58
PLK4 O00444 2/20 0.58
GAK O14976 2/20 0.58
RIPK2 O43353 2/20 0.58
ERN1 O75460 2/20 0.58
STK10 O94804 2/20 0.58
FYN P06241 2/20 0.58
YES1 P07947 2/20 0.58
LYN P07948 2/20 0.58
MET P08581 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15084515 0.94 KDR (0.66) KDRFLT4AURKBPDGFRBTEK
SCHEMBL15084560 0.94 KDR (0.66) KDRFLT4AURKBPDGFRBTEK
SCHEMBL15084599 0.93 ABCB11 (0.67) KDRFLT4AURKBPDGFRBTEK
SCHEMBL2744735 0.91 AXL (0.78) KDRFLT4AURKBPDGFRBTEK
SCHEMBL30001610 0.91 AXL (0.78) KDRFLT4AURKBPDGFRBTEK
SCHEMBL15084619 0.91 AXL (0.78) KDRFLT4AURKBPDGFRBTEK
SCHEMBL4031626 0.89 KDR (0.70) KDRFLT4AURKBPDGFRBTEK
SCHEMBL5570163 0.88 AXL (0.73) KDRFLT4AURKBPDGFRBTEK
SCHEMBL698905 0.87 AXL (0.84) KDRAURKBPDGFRBAURKAAXL
SCHEMBL29631712 0.86 AXL (0.71) KDRFLT4AURKBPDGFRBTEK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013097753-A1 FUSED HETEROCYCLIC DERIVATIVE AND APPLICATION THEREOF 江苏先声药业有限公司 (CN) 2013-07-04 WO disclosed