SCHEMBL15095491

SCHEMBL15095491

CNc1ccc(O)c(-c2ccnn2C)c1

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.50
MAPT P10636 1/20 0.50
HTR2A P28223 15/20 0.43
HTR2C P28335 13/20 0.43
KDM4C Q9H3R0 2/20 0.40
COMT P21964 1/20 0.40
IDO1 P14902 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2064347 0.82 KDM4C (0.51) ALDH1A1MAPTHTR2AHTR2CKDM4C
SCHEMBL19442038 0.82 ALDH1A1 (0.46) ALDH1A1MAPTHTR2AHTR2CKDM4C
SCHEMBL364560 0.81 MAPT (0.65) ALDH1A1MAPTHTR2AHTR2CCOMT
SCHEMBL13144356 0.79 MAPT (0.50) ALDH1A1MAPTCOMTIDO1
SCHEMBL2064569 0.78 MAPT (0.49) ALDH1A1MAPTHTR2AHTR2CKDM4C
SCHEMBL323525 0.78 MAPT (0.49) ALDH1A1MAPTCOMTIDO1
SCHEMBL1095146 0.78 ALDH1A1 (0.49) ALDH1A1MAPTHTR2AHTR2CCOMT
SCHEMBL29573491 0.77 HTR2A (0.73) HTR2AHTR2C
SCHEMBL1166246 0.77 HTR2A (0.73) HTR2AHTR2C
SCHEMBL16705330 0.75 MAPT (0.47) ALDH1A1MAPTKDM4CCOMTIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8481535-B2 Crystalline forms and processes for the preparation of phenyl-pyrazoles useful as modulators of the 5-HT2A serotonin receptor ARENA PHARMACEUTICALS, INC. (US) 2013-07-09 US disclosed