SCHEMBL1509722

SCHEMBL1509722

COc1ncccc1-c1ccc(O)c(-c2nc3cc(C(=O)Nc4ccc(CCN5CCC6(CC5)NC(=O)N(C)C6=O)cc4)ccc3[nH]2)c1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 6/20 0.41
ABCB1 P08183 5/20 0.41
HPSE Q9Y251 9/20 0.38
GSK3B P49841 1/20 0.36
CARM1 Q86X55 1/20 0.36
ADORA2A P29274 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1509427 0.91 ABCG2 (0.40) ABCG2ABCB1HPSEGSK3BCARM1
SCHEMBL12834002 0.89 ABCB1 (0.45) ABCG2ABCB1HPSEGSK3BCARM1
SCHEMBL1509459 0.88 ABCG2 (0.42) ABCG2ABCB1HPSEGSK3BADORA2A
SCHEMBL12833550 0.88 ABCB1 (0.44) ABCG2ABCB1HPSEGSK3BCARM1
SCHEMBL14090449 0.88 ABCG2 (0.44) ABCG2ABCB1HPSEGSK3BCARM1
SCHEMBL12833673 0.87 ABCB1 (0.43) ABCG2ABCB1HPSEADORA2A
SCHEMBL1509641 0.86 DRD2 (0.43) ABCG2ABCB1HPSEGSK3BADORA2A
SCHEMBL14090443 0.86 ABCB1 (0.43) ABCG2ABCB1HPSEGSK3BCARM1
SCHEMBL1509498 0.84 ABCG2 (0.48) ABCG2ABCB1HPSECARM1
SCHEMBL14090416 0.83 DDR2 (0.49) HPSE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2298770-A1 Heterocyclic compounds as TrkA modulators ChemBridge Corporation (US) 2011-03-23 EP disclosed