SCHEMBL15099404

SCHEMBL15099404

CN1CCC2(CC1)CC(c1ccccc1)C(=O)N2C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.44
KMT2A Q03164 1/20 0.44
SIGMAR1 Q99720 5/20 0.40
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
CHRM1 P11229 1/20 0.38
KDM1A O60341 1/20 0.37
HTR2A P28223 2/20 0.37
HTR2C P28335 2/20 0.37
HTR2B P41595 2/20 0.37
DRD2 P14416 1/20 0.37
MAPK1 P28482 1/20 0.36
THPO P40225 1/20 0.36
HIF1A Q16665 1/20 0.36
HSD17B10 Q99714 1/20 0.36
DRD1 P21728 1/20 0.36
MTOR P42345 1/20 0.36
GRM5 P41594 1/20 0.36
DRD4 P21917 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9965993 0.72 KMT2A (0.46) TSHRKMT2ASIGMAR1SLC6A2SLC6A4
SCHEMBL15099393 0.72 CHRM2 (0.41) TSHRKMT2ASIGMAR1SLC6A2SLC6A4
SCHEMBL16203621 0.65 TSHR (0.53) TSHRKMT2ACHRM1DRD2GRM5
SCHEMBL15203830 0.65 TSHR (0.53) TSHRKMT2ACHRM1DRD2GRM5
SCHEMBL15099412 0.65 AGTR2 (0.47) TSHRKMT2ASIGMAR1CHRM1KDM1A
SCHEMBL11618119 0.64 SLC6A2 (0.53) TSHRKMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL27262808 0.64 TSHR (0.56) TSHRKMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL12932720 0.64 CHRM1 (0.41) TSHRSIGMAR1CHRM1KDM1AHTR2A
SCHEMBL16356788 0.63 AGTR2 (0.49) TSHRSIGMAR1CHRM1KDM1AHTR2A
SCHEMBL11275319 0.63 CHRM1 (0.43) TSHRKMT2ASIGMAR1CHRM1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013102242-A1 HETEROCYCLIC COMPOUNDS AND METHODS FOR THEIR USE SPINIFEX PHARMACEUTICALS PTY LTD (AU) 2013-07-11 WO disclosed