SCHEMBL15211634

SCHEMBL15211634

CCc1cc(OCc2ccc(C)nc2C)cc2scc(OC(C)=O)c12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 5/20 0.36
PPARA Q07869 5/20 0.36
MAPT P10636 3/20 0.33
LMNA P02545 2/20 0.33
HTT P42858 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
MAPK1 P28482 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PPARG P37231 1/20 0.33
ADK P55263 1/20 0.33
ADORA2A P29274 2/20 0.32
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17431435 0.93 PPARD (0.34) PPARDPPARAMAPTPPARGADK
SCHEMBL15211275 0.91 PPARD (0.39) PPARDPPARAMAPTKDM4EALDH1A1
SCHEMBL15211344 0.89 PPARD (0.42) PPARDPPARAMAPTLMNAHTT
SCHEMBL15211745 0.89 POLB (0.35) PPARDPPARAMAPTALDH1A1GLA
SCHEMBL15211256 0.89 PPARD (0.35) PPARDPPARAPPARGADKNPC1
SCHEMBL15211484 0.87 PPARD (0.33) PPARDPPARAPPARGADKPDE10A
SCHEMBL15211568 0.87 PPARD (0.33) PPARDPPARALMNAHTTPPARG
SCHEMBL15211299 0.86 PPARD (0.39) PPARDPPARAPPARGADK
SCHEMBL15211438 0.86 PPARD (0.34) PPARDPPARAPPARGADK
SCHEMBL15211293 0.86 IKBKB (0.34) PPARDPPARAMAPTLMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9238639-B2 Aromatic ring compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-01-19 US disclosed
EP-2838891-A1 AROMATIC RING COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-02-25 EP disclosed
WO-2013125732-A1 AROMATIC RING COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-08-29 WO disclosed