SCHEMBL15214059

SCHEMBL15214059

Cc1ccc(-c2nnco2)cc1-c1cnc(NC(=O)c2snnc2C)cn1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
IL2 P60568 11/20 0.46
LMNA P02545 1/20 0.39
CREBBP Q92793 1/20 0.39
POLB P06746 1/20 0.37
USP2 O75604 1/20 0.36
RAF1 P04049 2/20 0.36
BRAF P15056 2/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15214062 0.91 POLB (0.42) IL2LMNACREBBPPOLBUSP2
SCHEMBL8259711 0.87 IL2 (0.46) IL2LMNAPOLBUSP2KDM4E
SCHEMBL15214063 0.85 IL2 (0.44) IL2LMNAPOLB
SCHEMBL17435148 0.85 IL2 (0.40) IL2LMNACREBBPPOLBUSP2
SCHEMBL15214060 0.83 IL2 (0.43) IL2LMNAPOLB
SCHEMBL15214066 0.82 IL2 (0.46) IL2LMNAPOLBUSP2KDM4E
SCHEMBL15214067 0.81 IL2 (0.45) IL2LMNAPOLBUSP2KDM4E
SCHEMBL15942556 0.81 IL2 (0.49) IL2LMNACREBBPPOLBUSP2
SCHEMBL15214064 0.81 IL2 (0.43) IL2LMNAPOLBUSP2KDM4E
SCHEMBL5550955 0.81 IL2 (0.64) IL2CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9493427-B2 Compounds for inflammation and immune-related uses SYNTA PHARMACEUTICALS CORP. (US) 2016-11-15 US disclosed
EP-1848435-B1 COMPOUNDS AGAINST INFLAMMATIONS AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP (US) 2016-01-20 EP disclosed
US-20150266829-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES PRCL Research Inc. (CA) 2015-09-24 US disclosed
US-20150266829-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES PRCL Research Inc. (CA) 2015-09-24 US disclosed
US-9090570-B2 Compounds for inflammation and immune-related uses PRCL Research Inc. (CA) 2015-07-28 US disclosed
US-8518950-B2 pyrazinyl, pyrimidinyl and pyridazinyl derivatives such asN-[5-(2-Chloro-5-trifluoromethyl-phenyl)-pyrazin-2-yl]-2,6-difluoro-benzamide, used as immunosuppressants for the treatmet or prevent inflammatory and immune disorders SYNTA PHARMACEUTICALS CORP. (US) 2013-08-27 US disclosed
US-8518950-B2 pyrazinyl, pyrimidinyl and pyridazinyl derivatives such asN-[5-(2-Chloro-5-trifluoromethyl-phenyl)-pyrazin-2-yl]-2,6-difluoro-benzamide, used as immunosuppressants for the treatmet or prevent inflammatory and immune disorders SYNTA PHARMACEUTICALS CORP. (US) 2013-08-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150266829-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES CCR1, CCR9, CXCR2 IL2 21/4885LMNA 3271/4885CREBBP 1789/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.