SCHEMBL15214201

SCHEMBL15214201

CCCCCCCCCCCCCCCCCCCC(=O)n1c2ncnc3c(ncn3C(=O)CCCCCCCCCCCCC)c-2nc1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.37
SQOR Q9Y6N5 2/20 0.35
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32
OXER1 Q8TDS5 7/20 0.32
ADA P00813 4/20 0.32
PDE2A O00408 3/20 0.32
CYP3A4 P08684 2/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12112267 1.00 GSK3B (0.37) GSK3BSQORPSEN1PSEN2APH1B
SCHEMBL15214190 0.88 ADA (0.36) GSK3BADAPDE2ACYP3A4PDE4A
SCHEMBL12112264 0.87 PDE4A (0.36) GSK3BSQORPDE4APDE4BPDE4C
SCHEMBL28863078 0.77 GSK3B (0.63) GSK3BADAPDE2ACYP3A4PDE4A
SCHEMBL5468657 0.77 GSK3B (0.63) GSK3BADAPDE2ACYP3A4PDE4A
SCHEMBL29601253 0.69 HDAC1 (0.44) GSK3BSQOROXER1ALDH1A1LMNA
SCHEMBL29601213 0.69 HDAC1 (0.42) GSK3BSQOR
SCHEMBL15214197 0.68 ADORA2A (0.49) KDM4EALDH1A1CYP1A2HSD17B10TSHR
SCHEMBL5347874 0.68 PNP (0.50) SQORHSD17B10TSHRBLM
SCHEMBL12112263 0.68 ADORA2A (0.49) KDM4EALDH1A1CYP1A2HSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8518901-B2 Fused diimidazodiazepine compounds and methods of use and manufacture thereof THE JOHNS HOPKINS UNIVERSITY (US) 2013-08-27 US disclosed