SCHEMBL15218451

SCHEMBL15218451

CS(=O)(=O)Nc1ccc(Cl)c(C(F)(F)F)c1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.57
KMT2A Q03164 2/20 0.56
MAPT P10636 2/20 0.54
TP53 P04637 1/20 0.54
KIF11 P52732 2/20 0.54
CYP17A1 P05093 3/20 0.52
RAPGEF4 Q8WZA2 1/20 0.51
PDK1 Q15118 1/20 0.51
CA1 P00915 3/20 0.51
CA2 P00918 3/20 0.51
CA7 P43166 3/20 0.51
CA9 Q16790 3/20 0.51
CNR2 P34972 1/20 0.51
EPHX2 P34913 1/20 0.48
NR1H4 Q96RI1 1/20 0.48
CCR2 P41597 1/20 0.48
LMNA P02545 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13145697 0.86 HPGD (0.49) MAPTKIF11CYP17A1EPHX2NR1H4
SCHEMBL3377569 0.86 KIF11 (0.51) KDRKMT2AMAPTTP53KIF11
SCHEMBL15220225 0.81 CYP17A1 (0.60) KIF11CYP17A1
SCHEMBL3375785 0.81 KIF11 (0.59) MAPTKIF11CYP17A1
SCHEMBL10804574 0.81 MAPT (0.69) KMT2AMAPTTP53CA1CA2
SCHEMBL527332 0.80 KIF11 (0.54) KMT2AMAPTKIF11CYP17A1CA1
SCHEMBL22060018 0.80 KIF11 (0.57) MAPTKIF11CYP17A1
SCHEMBL9390760 0.78 HPGD (0.58) KIF11CYP17A1EPHX2LMNA
SCHEMBL31240769 0.78 KIF11 (0.51) KMT2AKIF11CYP17A1EPHX2NR1H4
SCHEMBL3932771 0.77 KIF11 (0.50) KMT2AMAPTKIF11CYP17A1RAPGEF4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3323813-A1 HISTONE ACETYLTRANSFERASE MODULATORS AND USES THEREOF The Trustees of Columbia University in the City of New York (US) 2018-05-23 EP disclosed
US-20170121276-A1 HISTONE ACETYLTRANSFERASE MODULATORS AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2017-05-04 US disclosed
US-9274419-B2 Blue photosensitive resin composition for color filter and application thereof CHI MEI CORPORATION (TW) 2016-03-01 US disclosed
US-20150268554-A1 BLUE PHOTOSENSITIVE RESIN COMPOSITION FOR COLOR FILTER AND APPLICATION THEREOF CHI MEI CORPORATION (TW) 2015-09-24 US disclosed
US-9086532-B2 Blue photosensitive resin composition for color filter and uses thereof CHI MEI CORPORATION (TW) 2015-07-21 US disclosed
US-9081142-B2 Photosensitive resin composition for a color filter and uses thereof CHI MEI CORPORATION (TW) 2015-07-14 US disclosed
US-20150042931-A1 BLUE PHOTOSENSITIVE RESIN COMPOSITION FOR COLOR FILTER AND USES THEREOF CHI MEI CORPORATION (TW) 2015-02-12 US disclosed
US-20140346416-A1 PHOTOSENSITIVE RESIN COMPOSITION FOR A COLOR FILTER AND USES THEREOF CHI MEI CORPORATION (TW) 2014-11-27 US disclosed
US-20130222738-A1 COLOR LIQUID CRYSTAL DISPLAY DEVICE CHI MEI CORPORATION (TW) 2013-08-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170121276-A1 HISTONE ACETYLTRANSFERASE MODULATORS AND USES THEREOF EP300, KAT2A, HTT KDR 4841/4885KMT2A 51/4885MAPT 8/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.