SCHEMBL1521987

SCHEMBL1521987

CCN1C(=O)N(c2ccc(F)c(NC(=O)NC3CCCCC3)c2)Cc2cnc(NC)cc21

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 8/20 0.43
FGFR4 P22455 8/20 0.43
PARP1 P09874 1/20 0.40
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
KMT2A Q03164 2/20 0.39
EPHX2 P34913 3/20 0.39
POLB P06746 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
FGFR2 P21802 2/20 0.35
FGFR3 P22607 2/20 0.35
KIT P10721 1/20 0.35
PDGFRA P16234 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1521947 0.90 RAB9A (0.41) PARP1NPC1RAB9AKMT2AEPHX2
SCHEMBL29894322 0.88 NPC1 (0.40) FGFR1FGFR4PARP1NPC1RAB9A
SCHEMBL1521769 0.88 NPC1 (0.40) FGFR1FGFR4PARP1NPC1RAB9A
SCHEMBL1522057 0.88 NPC1 (0.39) PARP1NPC1RAB9AKMT2AEPHX2
SCHEMBL1521844 0.88 FGFR1 (0.42) FGFR1FGFR4PARP1NPC1RAB9A
SCHEMBL1521676 0.86 PARP1 (0.38) PARP1NPC1RAB9AKMT2AEPHX2
SCHEMBL1521817 0.84 BRAF (0.40) FGFR1FGFR4KMT2AKITPDGFRA
SCHEMBL1521812 0.82 KIT (0.40) FGFR1FGFR4RAB9AKMT2AFGFR2
SCHEMBL1521600 0.81 KRAS (0.37) FGFR1FGFR4FGFR2FGFR3KIT
SCHEMBL1521807 0.80 MAPK14 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110118271-A1 Kinase Inhibitors Useful For The Treatment Of Proliferative Diseases FLYNN DANIEL L 2011-05-19 US claimed
US-7897762-B2 Kinase inhibitors useful for the treatment of proliferative diseases DECIPHERA PHARMACEUTICALS, LLC (US) 2011-03-01 US claimed
US-20090099190-A1 Kinase inhibitors useful for the treatment of proliferative diseases DECIPHERA PHARMACEUTICALS, LLC (US) 2009-04-16 US claimed
US-20110118271-A1 Kinase Inhibitors Useful For The Treatment Of Proliferative Diseases FLYNN DANIEL L 2011-05-19 US disclosed
US-7897762-B2 Kinase inhibitors useful for the treatment of proliferative diseases DECIPHERA PHARMACEUTICALS, LLC (US) 2011-03-01 US disclosed
US-20090099190-A1 Kinase inhibitors useful for the treatment of proliferative diseases DECIPHERA PHARMACEUTICALS, LLC (US) 2009-04-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110118271-A1 Kinase Inhibitors Useful For The Treatment Of Proliferative Diseases BRAF, PRKDC, RAF1 FGFR1 577/4885FGFR4 1073/4885PARP1 392/4885
US-20090099190-A1 Kinase inhibitors useful for the treatment of proliferative diseases BRAF, PRKDC, RAF1 FGFR1 577/4885FGFR4 1073/4885PARP1 392/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.