SCHEMBL1523038

SCHEMBL1523038

CC(C)CCn1c(=O)c(C2=NS(O)(O)c3cc(OC(C(=O)O)C(C)(C)C)ccc3N2)c(O)c2cccnc21

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP2C9 P11712 3/20 0.40
RXFP1 Q9HBX9 6/20 0.36
THRB P10828 1/20 0.36
MAPT P10636 5/20 0.36
TP53 P04637 2/20 0.35
NR1I2 O75469 1/20 0.32
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
HTR3A P46098 1/20 0.32
HTR3D Q70Z44 1/20 0.32
HTR3C Q8WXA8 1/20 0.32
PPARG P37231 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1523042 0.93 CYP2C9 (0.47) MAPK1HSD17B10CYP2C9RXFP1THRB
SCHEMBL1523423 0.88 CYP2C9 (0.41) MAPK1HSD17B10CYP2C9RXFP1THRB
SCHEMBL1522560 0.88 MAPK1 (0.42) MAPK1HSD17B10CYP2C9RXFP1THRB
SCHEMBL1522569 0.88 MAPK1 (0.41) MAPK1HSD17B10CYP2C9RXFP1THRB
SCHEMBL1522457 0.87 MAPK1 (0.42) MAPK1HSD17B10CYP2C9RXFP1THRB
SCHEMBL1522828 0.87 MAPK1 (0.41) MAPK1HSD17B10CYP2C9RXFP1THRB
SCHEMBL1522703 0.86 CYP2C9 (0.48) MAPK1HSD17B10CYP2C9RXFP1THRB
SCHEMBL1523324 0.86 MAPK1 (0.41) MAPK1HSD17B10CYP2C9RXFP1THRB
SCHEMBL1523725 0.86 MAPK1 (0.41) MAPK1HSD17B10CYP2C9RXFP1THRB
SCHEMBL1522877 0.86 MAPK1 (0.41) MAPK1HSD17B10CYP2C9RXFP1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7902203-B2 Anti-infective agents ABBOTT LABORATORIES, INC. (US) 2011-03-08 US disclosed