SCHEMBL1523042

SCHEMBL1523042

CC(C)CCn1c(=O)c(C2=NS(=O)(=O)c3cc(OC(C(=O)O)C(C)(C)C)ccc3N2)c(O)c2cccnc21

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.47
MAPK1 P28482 1/20 0.47
HSD17B10 Q99714 1/20 0.47
NR1I2 O75469 1/20 0.38
RXFP1 Q9HBX9 6/20 0.36
THRB P10828 1/20 0.36
MAPT P10636 5/20 0.36
TP53 P04637 2/20 0.35
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
HTR3A P46098 1/20 0.32
HTR3D Q70Z44 1/20 0.32
HTR3C Q8WXA8 1/20 0.32
PPARG P37231 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1523038 0.93 MAPK1 (0.40) CYP2C9MAPK1HSD17B10NR1I2RXFP1
SCHEMBL1523427 0.88 CYP2C9 (0.48) CYP2C9MAPK1HSD17B10NR1I2RXFP1
SCHEMBL1522557 0.88 MAPK1 (0.50) CYP2C9MAPK1HSD17B10NR1I2RXFP1
SCHEMBL7077611 0.88 CYP2C9 (0.59) CYP2C9MAPK1HSD17B10NR1I2RXFP1
SCHEMBL1522570 0.88 MAPK1 (0.48) CYP2C9MAPK1HSD17B10NR1I2RXFP1
SCHEMBL1522456 0.87 MAPK1 (0.49) CYP2C9MAPK1HSD17B10NR1I2RXFP1
SCHEMBL1522826 0.87 MAPK1 (0.49) CYP2C9MAPK1HSD17B10NR1I2RXFP1
SCHEMBL1523325 0.86 MAPK1 (0.49) CYP2C9MAPK1HSD17B10NR1I2RXFP1
SCHEMBL1522705 0.86 CYP2C9 (0.56) CYP2C9MAPK1HSD17B10NR1I2RXFP1
SCHEMBL1522875 0.86 MAPK1 (0.48) CYP2C9MAPK1HSD17B10NR1I2RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2361913-A1 Anti-infective agents Abbott Laboratories (US) 2011-08-31 EP disclosed
US-7902203-B2 Anti-infective agents ABBOTT LABORATORIES, INC. (US) 2011-03-08 US disclosed