SCHEMBL15310337

SCHEMBL15310337

O=C(c1ccc(-c2ccc(F)cc2F)cc1)C1CC2CCC(c3ncccn3)(C1)N2

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
F10 P00742 1/20 0.36
ACKR3 P25106 6/20 0.35
MGLL Q99685 1/20 0.35
AKT1 P31749 1/20 0.34
KLKB1 P03952 3/20 0.34
APP P05067 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
CYP2D6 P10635 1/20 0.34
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
PDE4B Q07343 1/20 0.33
HTR2A P28223 1/20 0.33
DYRK1A Q13627 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3577929 0.73 SLC6A7 (0.41) F10KLKB1ALDH1A1LMNAHTT
SCHEMBL14160624 0.68 TDP1 (0.41) ALDH1A1LMNAHTTHTR2A
SCHEMBL3577425 0.64 MAPK1 (0.43) ALDH1A1LMNAHTT
SCHEMBL411705 0.61 BCL2L1 (0.62) APPCYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL3585870 0.61 SLC6A7 (0.76) ALDH1A1
SCHEMBL18503388 0.61 MEN1 (0.47) CYP2D6ALDH1A1
SCHEMBL30747689 0.60 MAOB (0.55) APPCYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL10436026 0.60 MAOB (0.55) APPCYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL18924450 0.58 MAPK14 (0.58) ALDH1A1
SCHEMBL18503386 0.58 MEN1 (0.47) CYP2D6ALDH1A1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893212-B1 MULTICYCLIC COMPOUNDS AND METHODS OF THEIR USE LEXICON PHARMACEUTICALS INC (US) 2013-10-16 EP disclosed