SCHEMBL15310564

SCHEMBL15310564

CCOC(=O)C(C)(CCCc1ccc(Oc2cccc(C(F)(F)F)c2)cc1Cl)NC(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
PPARG P37231 6/20 0.38
PPARD Q03181 5/20 0.38
PPARA Q07869 5/20 0.38
FAAH O00519 2/20 0.36
THRB P10828 1/20 0.36
EGFR P00533 1/20 0.36
ERBB2 P04626 1/20 0.36
SCN9A Q15858 1/20 0.36
HTR2A P28223 1/20 0.36
SLC6A4 P31645 1/20 0.36
KCNH2 Q12809 1/20 0.36
KDM4E B2RXH2 3/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MRGPRX4 Q96LA9 1/20 0.35
GHSR Q92847 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3299440 1.00 TLR8 (0.38) TLR8TLR7PPARGPPARDPPARA
SCHEMBL3574671 0.90 TLR8 (0.40) TLR8TLR7PPARGPPARDPPARA
SCHEMBL3574667 0.90 TLR8 (0.40) TLR8TLR7PPARGPPARDPPARA
SCHEMBL3299890 0.85 TLR8 (0.41) TLR8TLR7PPARGPPARDPPARA
SCHEMBL3299897 0.85 TLR8 (0.41) TLR8TLR7PPARGPPARDPPARA
SCHEMBL3308752 0.82 TLR8 (0.42) TLR8TLR7PPARGPPARDPPARA
SCHEMBL3308747 0.82 TLR8 (0.42) TLR8TLR7PPARGPPARDPPARA
SCHEMBL15310409 0.80 SIRT2 (0.37) THRBSLC6A4KDM4ENPSR1MRGPRX4
SCHEMBL3301977 0.80 SIRT2 (0.37) THRBSLC6A4KDM4ENPSR1MRGPRX4
SCHEMBL1455821 0.80 THRB (0.41) THRBKDM4ENPSR1SMN1; SMN2MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058317-B1 AMINOPHOSPHORIC ACID ESTER DERIVATIVE AND S1P RECEPTOR MODULATOR CONTAINING THE SAME AS ACTIVE INGREDIENT KYORIN SEIYAKU KK (JP) 2013-10-16 EP disclosed