SCHEMBL15310658

SCHEMBL15310658

COC(=O)C(C)(C)[C@H]1C[C@H](N(C)C)CC[C@@H]1N1CCC(NC(=O)c2cccc(C(F)(F)F)c2)C1=O

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 20/20 0.61
CCR5 P51681 4/20 0.61
KCNH2 Q12809 5/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15310659 0.87 CCR2 (0.61) CCR2CCR5KCNH2
SCHEMBL3734010 0.86 CCR2 (0.66) CCR2CCR5KCNH2
SCHEMBL3734008 0.85 CCR2 (0.65) CCR2CCR5KCNH2
SCHEMBL3733046 0.83 CCR2 (0.70) CCR2CCR5KCNH2
SCHEMBL3733041 0.83 CCR2 (0.70) CCR2CCR5KCNH2
SCHEMBL3733051 0.83 CCR2 (0.70) CCR2CCR5KCNH2
SCHEMBL15310601 0.83 CCR2 (0.68) CCR2CCR5KCNH2
SCHEMBL3739574 0.82 CCR2 (0.77) CCR2CCR5KCNH2
SCHEMBL3739577 0.82 CCR2 (0.77) CCR2CCR5KCNH2
SCHEMBL3739567 0.82 CCR2 (0.77) CCR2CCR5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656345-B1 CYCLIC DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL MYERS SQUIBB CO (US) 2013-10-16 EP disclosed