SCHEMBL15313629

SCHEMBL15313629

Cc1ccc(-c2nc3n(c2Nc2ccc(F)c(F)c2)CCN(C(=O)C(C)(C)N)C3)cc1

nearest known ligand 0.88

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.88
CYP3A4 P08684 1/20 0.38
TP53 P04637 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
TACR3 P29371 1/20 0.36
CSNK1E P49674 3/20 0.35
P2RX7 Q99572 1/20 0.35
CSNK1D P48730 2/20 0.35
PDK2 Q15119 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2068306 0.95 KCNH2 (0.82) KCNH2CYP3A4TACR3CSNK1EP2RX7
SCHEMBL999379 0.94 KCNH2 (1.00) KCNH2CYP3A4CSNK1EP2RX7CSNK1D
SCHEMBL2068840 0.90 KCNH2 (0.80) KCNH2CYP3A4TP53GAAMAPT
SCHEMBL2068261 0.90 KCNH2 (1.00) KCNH2CYP3A4TP53CSNK1ECSNK1D
SCHEMBL1000956 0.89 KCNH2 (0.87) KCNH2CYP3A4CSNK1EP2RX7CSNK1D
SCHEMBL1044397 0.89 KCNH2 (0.87) KCNH2CYP3A4CSNK1ECSNK1DPDK2
SCHEMBL1050937 0.87 KCNH2 (0.80) KCNH2CYP3A4TACR3CSNK1EP2RX7
SCHEMBL12781873 0.86 KCNH2 (0.82) KCNH2CYP3A4GAAMAPTPDK2
SCHEMBL2069758 0.86 KCNH2 (1.00) KCNH2CYP3A4TACR3CSNK1EP2RX7
SCHEMBL2069186 0.86 KCNH2 (0.84) KCNH2CYP3A4MAPTP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9469645-B2 Compounds and compositions for the treatment of parasitic diseases NOVARTIS AG (CH) 2016-10-18 US disclosed
US-20130281403-A1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF PARASITIC DISEASES IRM LLC (BM) 2013-10-24 US disclosed
US-8557801-B2 Compounds and compositions useful for the treatment of parasitic diseases IRM LLC (BM) 2013-10-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130281403-A1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF PARASITIC DISEASES SQLE, ABCB1, FDPS KCNH2 1679/4885CYP3A4 97/4885TP53 4077/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.