SCHEMBL15313666

SCHEMBL15313666

COc1c(C(=O)O)cc(S(=O)(=O)Cl)c(OC)c1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.46
KDM4E B2RXH2 4/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ALDH1A1 P00352 3/20 0.39
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA3 P07451 2/20 0.39
CA4 P22748 2/20 0.39
CA6 P23280 2/20 0.39
CA5A P35218 2/20 0.39
CA7 P43166 2/20 0.39
CA9 Q16790 2/20 0.39
CA13 Q8N1Q1 2/20 0.39
CA14 Q9ULX7 2/20 0.39
CA5B Q9Y2D0 2/20 0.39
TRPV4 Q9HBA0 1/20 0.39
HPGD P15428 1/20 0.39
MAPT P10636 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9110910 0.81 MCL1 (0.54) HSD17B10KDM4ENPSR1ALDH1A1HPGD
SCHEMBL11267450 0.79 KDM4E (0.39) HSD17B10KDM4ENPSR1ALDH1A1CA12
SCHEMBL7801303 0.77 KDM4E (0.63) HSD17B10KDM4ENPSR1ALDH1A1CA12
SCHEMBL2004907 0.76 F2 (0.47) HSD17B10KDM4EALDH1A1CA1CA2
SCHEMBL27859515 0.76 TPMT (0.53) HSD17B10KDM4EALDH1A1HPGDMAPT
SCHEMBL9056913 0.75 CYP1A1 (0.49) HSD17B10KDM4EALDH1A1HPGDMAPT
SCHEMBL10721874 0.75 KDM4E (0.52) HSD17B10KDM4ENPSR1ALDH1A1CA12
SCHEMBL4905793 0.75 NPSR1 (0.49) HSD17B10KDM4ENPSR1ALDH1A1CA12
SCHEMBL11005985 0.75 CA1 (0.47) HSD17B10KDM4ENPSR1ALDH1A1CA12
SCHEMBL8846922 0.75 KDM4E (0.52) HSD17B10KDM4ENPSR1ALDH1A1TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8557812-B2 Small molecule inhibitors of anti-apoptotic BCL-2 family members and the uses thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2013-10-15 US disclosed
US-8557812-B2 Small molecule inhibitors of anti-apoptotic BCL-2 family members and the uses thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2013-10-15 US disclosed