SCHEMBL15324072

SCHEMBL15324072

COc1ccnc(C2=C[C]=CCN2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.54
CCR5 P51681 1/20 0.54
CCR8 P51685 1/20 0.54
NOS3 P29474 2/20 0.40
NOS1 P29475 2/20 0.40
NOS2 P35228 2/20 0.40
PLAU P00749 1/20 0.38
SYK P43405 6/20 0.37
CBFB Q13951 2/20 0.36
DYRK1A Q13627 4/20 0.34
NISCH Q9Y2I1 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2D6 P10635 2/20 0.34
KDM4E B2RXH2 1/20 0.34
DYRK3 O43781 1/20 0.34
CCNT1 O60563 1/20 0.34
CCNB2 O95067 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CDK1 P06493 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15322772 0.80 CCR1 (0.50) CCR1CCR5CCR8NOS3NOS1
SCHEMBL8738510 0.73 CCR1 (0.54) CCR1CCR5CCR8NOS3NOS1
SCHEMBL182529 0.73 CCR1 (1.00) CCR1CCR5CCR8NOS3NOS1
SCHEMBL29395249 0.73 CCR1 (1.00) CCR1CCR5CCR8NOS3NOS1
SCHEMBL4656344 0.71 KDM4E (0.45) CCR1CCR5CCR8NISCHCYP1A2
Hydrochloric Acid SCHEMBL29903189 0.71 CCR1 (0.95) CCR1CCR5CCR8NOS3NOS1
SCHEMBL28212407 0.71 CCR1 (0.95) CCR1CCR5CCR8NOS3NOS1
SCHEMBL9135460 0.71 CCR1 (0.95) CCR1CCR5CCR8NOS3NOS1
Methane SCHEMBL21386924 0.71 CCR1 (0.95) CCR1CCR5CCR8NOS3NOS1
SCHEMBL8746042 0.71 CCR1 (0.95) CCR1CCR5CCR8NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2838534-A2 SUBSTITUTED BENZAMIDES AND THEIR USES The Board of Trustees of The Leland Stanford Junior University (US) 2015-02-25 EP disclosed
WO-2013155338-A2 SUBSTITUTED BENZAMIDES AND THEIR USES THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2013-10-17 WO disclosed