SCHEMBL15327433

SCHEMBL15327433

N#CCNC(=O)O[C@H]1C[C@@H](S(=O)(=O)c2ccccc2C(F)(F)F)CN1C(=O)C1CCCCC1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSS P25774 20/20 0.51
CTSL P07711 2/20 0.46
CTSB P07858 2/20 0.46
CTSK P43235 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15327529 0.92 CTSS (0.58) CTSSCTSLCTSBCTSK
SCHEMBL15327439 0.92 CTSS (0.52) CTSSCTSLCTSBCTSK
SCHEMBL15327241 0.88 CTSS (0.59) CTSSCTSLCTSB
SCHEMBL695748 0.87 CTSS (0.59) CTSSCTSLCTSBCTSK
SCHEMBL15327470 0.86 CTSS (0.52) CTSSCTSLCTSBCTSK
SCHEMBL15327267 0.85 CTSS (0.60) CTSSCTSLCTSB
SCHEMBL15327343 0.85 CTSS (0.49) CTSSCTSLCTSBCTSK
SCHEMBL15327612 0.84 CTSS (0.50) CTSSCTSLCTSBCTSK
SCHEMBL15327301 0.84 CTSS (0.50) CTSSCTSLCTSBCTSK
SCHEMBL15327492 0.84 CTSS (0.52) CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-B1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS HOFFMANN LA ROCHE (CH) 2013-10-23 EP claimed