SCHEMBL15327641

SCHEMBL15327641

CC(C)(C)OC(=O)ON1C[C@H](S(=O)(=O)c2ccc(N3CCC(F)(F)CC3)cc2Cl)C[C@H]1C(=O)NC1(C#N)CC1

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSS P25774 20/20 0.52
CTSL P07711 5/20 0.49
CTSB P07858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15327590 0.96 CTSS (0.51) CTSSCTSLCTSB
SCHEMBL15327344 0.93 CTSS (0.55) CTSSCTSLCTSB
SCHEMBL15327335 0.91 CTSS (0.52) CTSSCTSLCTSB
SCHEMBL15327365 0.90 CTSS (0.54) CTSSCTSLCTSB
SCHEMBL695616 0.88 CTSS (0.59) CTSSCTSLCTSB
SCHEMBL15327342 0.88 CTSS (0.56) CTSSCTSLCTSB
SCHEMBL15327566 0.87 CTSS (0.60) CTSSCTSLCTSB
SCHEMBL15327150 0.85 CTSS (0.61) CTSSCTSLCTSB
SCHEMBL15327368 0.84 CTSS (0.55) CTSSCTSLCTSB
SCHEMBL700242 0.84 CTSS (0.58) CTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-B1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS HOFFMANN LA ROCHE (CH) 2013-10-23 EP claimed