SCHEMBL15329626

SCHEMBL15329626

CNC(=O)C1CCN(c2ccc(C=O)o2)CC1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.63
POLB P06746 2/20 0.63
SMN1; SMN2 Q16637 2/20 0.55
RXFP1 Q9HBX9 1/20 0.41
CYP46A1 Q9Y6A2 1/20 0.40
F2 P00734 1/20 0.39
LTA4H P09960 1/20 0.38
NOTUM Q6P988 1/20 0.38
PDK2 Q15119 1/20 0.38
PIK3CA P42336 1/20 0.38
MAPT P10636 4/20 0.37
MEN1 O00255 4/20 0.37
KMT2A Q03164 4/20 0.37
USP2 O75604 3/20 0.37
IDE P14735 2/20 0.37
TNNI3 P19429 1/20 0.37
TNNT2 P45379 1/20 0.37
TNNC1 P63316 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2559210 0.82 ALDH1A1 (0.64) ALDH1A1POLBSMN1; SMN2F2MAPT
SCHEMBL1958069 0.78 ALDH1A1 (0.71) ALDH1A1POLBSMN1; SMN2F2MAPT
SCHEMBL15330523 0.76 ALDH1A1 (0.47) ALDH1A1POLBSMN1; SMN2PDK2PIK3CA
SCHEMBL15331610 0.75 POLB (0.48) ALDH1A1POLBSMN1; SMN2MAPTMEN1
SCHEMBL2560795 0.74 ALDH1A1 (0.61) ALDH1A1POLBSMN1; SMN2F2LTA4H
SCHEMBL2561051 0.73 TRIM24 (0.51) ALDH1A1SMN1; SMN2KDM4E
SCHEMBL15331289 0.72 CYP46A1 (0.53) ALDH1A1SMN1; SMN2RXFP1CYP46A1LTA4H
SCHEMBL20206188 0.70 POLB (0.63) ALDH1A1POLBSMN1; SMN2MAPTMEN1
SCHEMBL1960058 0.70 SMN1; SMN2 (0.73) ALDH1A1POLBSMN1; SMN2MAPTMEN1
SCHEMBL24713217 0.69 POLB (0.54) ALDH1A1POLBSMN1; SMN2MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-11225655-B2 Bi-functional complexes and methods for making and using such complexes NUEVOLUTION A/S (DK) 2022-01-18 US disclosed
EP-3540059-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2019-09-18 EP disclosed
EP-2558577-B1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION AS (DK) 2018-12-12 EP disclosed
US-20130281324-A1 BI-FUNCTINAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2013-10-24 US disclosed