SCHEMBL15375341

SCHEMBL15375341

C[C@H](O)[C@H](NC(=O)c1ccc(Cc2ccc(CN3CCOCC3)cc2)cc1)C(=O)NO

nearest known ligand 0.83

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.51
KMT2A Q03164 1/20 0.51
HIF1A Q16665 1/20 0.50
EPAS1 Q99814 1/20 0.50
MAPK1 P28482 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
RAB9A P51151 1/20 0.49
ALDH1A1 P00352 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13244853 1.00 NPC1 (0.51) NPC1KMT2AHIF1AEPAS1MAPK1
SCHEMBL15375340 1.00 NPC1 (0.51) NPC1KMT2AHIF1AEPAS1MAPK1
SCHEMBL3012101 1.00 NPC1 (0.51) NPC1KMT2AHIF1AEPAS1MAPK1
SCHEMBL1101249 0.97 NPC1 (0.54) NPC1KMT2AHIF1AEPAS1MAPK1
SCHEMBL9925870 0.94 KMT2A (0.51) NPC1KMT2AHIF1AEPAS1
SCHEMBL13267032 0.94 KDM4E (0.52) NPC1KMT2AHIF1AEPAS1ALDH1A1
SCHEMBL14400854 0.94 KMT2A (0.51) NPC1KMT2AHIF1AEPAS1
SCHEMBL13245569 0.94 KDM4E (0.52) NPC1KMT2AHIF1AEPAS1ALDH1A1
SCHEMBL1109224 0.94 KMT2A (0.51) NPC1KMT2AHIF1AEPAS1
SCHEMBL13267374 0.92 ALDH1A1 (0.50) NPC1KMT2AHIF1AEPAS1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2662353-A2 Antibacterial agents Achaogen, Inc. (US) 2013-11-13 EP disclosed