SCHEMBL15375593

SCHEMBL15375593

COC(=O)C(N)C(C)C(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA14 Q9ULX7 3/20 0.41
CA12 O43570 2/20 0.41
NOS1 P29475 2/20 0.39
NOS3 P29474 1/20 0.39
NOS2 P35228 1/20 0.39
DGAT1 O75907 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
LMNA P02545 1/20 0.30
KMT2A Q03164 1/20 0.30
CYP2D6 P10635 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15375592 1.00 CA14 (0.41) CA14CA12NOS1NOS3NOS2
Hydrochloric Acid SCHEMBL3023545 0.98 CA14 (0.40) CA14CA12NOS1NOS3NOS2
SCHEMBL3240752 0.85 NOS1 (0.41) CA14CA12NOS1NOS3NOS2
Hydrochloric Acid SCHEMBL28773975 0.83 NOS1 (0.41) CA14CA12NOS1NOS3NOS2
SCHEMBL13613724 0.83 CA14 (0.46) CA14CA12NOS1NOS3NOS2
SCHEMBL12281961 0.83 CA14 (0.46) CA14CA12NOS1NOS3NOS2
SCHEMBL15156959 0.83 SMN1; SMN2 (0.42) CA14CA12SMN1; SMN2CA1CA2
SCHEMBL28902221 0.83 SMN1; SMN2 (0.42) CA14CA12SMN1; SMN2CA1CA2
SCHEMBL27457895 0.82 SLC7A5 (0.44) CA14CA12NOS1NOS3NOS2
SCHEMBL15268524 0.79 NOS1 (0.39) CA14CA12NOS1NOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170814-B1 ANTIBACTERIAL AGENTS ACHAOGEN INC (US) 2016-08-17 EP disclosed
EP-2662353-A2 Antibacterial agents Achaogen, Inc. (US) 2013-11-13 EP disclosed