SCHEMBL15405418

SCHEMBL15405418

COc1c(OCCCN2CCOCC2)ccc2c(Oc3ccc(-c4cnc(Nc5ccc(F)cc5)n(C)c4=O)cc3F)ccnc12

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 18/20 0.79
MST1R Q04912 6/20 0.79
KDR P35968 5/20 0.79
RPS6KB1 P23443 4/20 0.79
TEK Q02763 4/20 0.79
BTK Q06187 4/20 0.79
HGF P14210 3/20 0.79
EGFR P00533 3/20 0.79
FLT4 P35916 3/20 0.79
JAK2 O60674 2/20 0.79
FLT1 P17948 2/20 0.79
FGFR2 P21802 2/20 0.79
AURKA O14965 3/20 0.60
LCK P06239 3/20 0.60
MAPK9 P45984 2/20 0.60
RPS6KA5 O75582 1/20 0.60
PIM1 P11309 1/20 0.60
CSF1R P07333 2/20 0.56
AXL P30530 3/20 0.49
PLK4 O00444 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15405203 0.95 MET (0.72) METMST1RKDRRPS6KB1TEK
SCHEMBL15404552 0.95 MET (0.71) METMST1RKDRRPS6KB1TEK
SCHEMBL15404511 0.95 MET (0.79) METMST1RKDRRPS6KB1TEK
SCHEMBL15405069 0.94 MET (0.70) METMST1RKDRRPS6KB1TEK
SCHEMBL15406338 0.89 MET (0.63) METMST1RKDRRPS6KB1TEK
SCHEMBL2868963 0.88 MET (1.00) METMST1RKDRRPS6KB1TEK
SCHEMBL29439859 0.88 MET (1.00) METMST1RKDRRPS6KB1TEK
SCHEMBL15405185 0.87 MET (0.77) METMST1RKDRRPS6KB1TEK
SCHEMBL2868521 0.84 MET (0.91) METMST1RKDRRPS6KB1TEK
SCHEMBL13511860 0.84 MET (0.91) METMST1RKDRRPS6KB1TEK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1827434-B1 QUINOLINES AND QUINAZOLINE ANALOGS AND THEIR USE AS MEDICAMENTS FOR TREATING CANCER AMGEN INC (US) 2014-01-15 EP claimed