SCHEMBL15414401

SCHEMBL15414401

CNC(C)C(=O)NC1CCc2ccccc2NC1=O

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PYGL P06737 2/20 0.57
PYGM P11217 2/20 0.57
XIAP P98170 13/20 0.53
RIPK1 Q13546 5/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25343594 0.88 PYGL (0.55) PYGLPYGMRIPK1
SCHEMBL25343601 0.88 PYGL (0.55) PYGLPYGMRIPK1
SCHEMBL15414842 0.88 PYGL (0.55) PYGLPYGMRIPK1
SCHEMBL17310767 0.86 PYGL (0.53) PYGLPYGMXIAPRIPK1
Hydrochloric Acid SCHEMBL25343578 0.85 PYGL (0.55) PYGLPYGMRIPK1
Hydrochloric Acid SCHEMBL25343581 0.85 PYGL (0.55) PYGLPYGMRIPK1
SCHEMBL29481025 0.82 PYGL (0.50) PYGLPYGMRIPK1
SCHEMBL4216634 0.80 PYGL (0.66) PYGLPYGMRIPK1
SCHEMBL1976547 0.80 PYGL (0.66) PYGLPYGMRIPK1
SCHEMBL4232147 0.80 PYGL (0.66) PYGLPYGMRIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2872490-A1 ANTIPROLIFERATIVE BENZO [B]AZEPIN- 2 - ONES F. Hoffmann-La Roche AG (CH) 2015-05-20 EP disclosed
WO-2014009495-A1 ANTIPROLIFERATIVE BENZO [B] AZEPIN- 2 - ONES F. HOFFMANN-LA ROCHE AG (CH) 2014-01-16 WO disclosed