SCHEMBL15417099

SCHEMBL15417099

Cc1cc(-c2cccn2C(=O)OC(C)(C)C)c(-c2cccn2C(=O)OC(C)(C)C)cc1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.53
HSP90AB1 P08238 1/20 0.53
PIK3R1 P27986 1/20 0.50
PIK3CA P42336 1/20 0.50
BUB1 O43683 1/20 0.43
TNK2 Q07912 1/20 0.41
BCHE P06276 1/20 0.40
ATR Q13535 1/20 0.38
MET P08581 1/20 0.37
AXL P30530 1/20 0.37
MERTK Q12866 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GPR119 Q8TDV5 2/20 0.34
LMNA P02545 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
NR1H2 P55055 2/20 0.34
CYP1A2 P05177 1/20 0.34
POLB P06746 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15417083 0.87 HSP90AA1 (0.52) HSP90AA1HSP90AB1PIK3R1PIK3CABUB1
SCHEMBL18812369 0.87 HSP90AA1 (0.49) HSP90AA1HSP90AB1PIK3R1PIK3CABUB1
SCHEMBL22036737 0.86 HSP90AA1 (0.53) HSP90AA1HSP90AB1PIK3R1PIK3CABUB1
SCHEMBL25594975 0.84 HSP90AA1 (0.53) HSP90AA1HSP90AB1PIK3R1PIK3CABUB1
SCHEMBL23306709 0.82 HSP90AA1 (0.51) HSP90AA1HSP90AB1PIK3R1PIK3CABUB1
SCHEMBL19953372 0.82 HSP90AA1 (0.51) HSP90AA1HSP90AB1PIK3R1PIK3CABUB1
SCHEMBL15498091 0.79 HSP90AA1 (0.54) HSP90AA1HSP90AB1PIK3R1PIK3CABUB1
SCHEMBL26819799 0.79 PIK3R1 (0.54) HSP90AA1HSP90AB1PIK3R1PIK3CABUB1
SCHEMBL24697208 0.79 HSP90AA1 (0.48) HSP90AA1HSP90AB1PIK3R1PIK3CABUB1
SCHEMBL30564364 0.79 PIK3R1 (0.51) HSP90AA1HSP90AB1PIK3R1PIK3CABUB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013183327-A1 METHOD FOR PRODUCING COMPOUND HAVING CONDENSED RING STRUCTURE, COMPOUND HAVING CONDENSED RING STRUCTURE, AND ORGANIC LIGHT-EMITTING DEVICE USING SAME 国立大学法人奈良先端科学技術大学院大学 (JP) 2013-12-12 WO disclosed