SCHEMBL15417529

SCHEMBL15417529

CCOC(=O)/C=C(\C)c1ccc(OC(F)F)c(OC(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 7/20 0.45
PDE4B Q07343 7/20 0.45
PDE4C Q08493 7/20 0.45
PDE4D Q08499 7/20 0.45
KDM4E B2RXH2 2/20 0.42
HTT P42858 2/20 0.42
RAB9A P51151 2/20 0.41
F2 P00734 1/20 0.41
PLG P00747 1/20 0.41
PRSS1 P07477 1/20 0.41
ALDH1A1 P00352 1/20 0.40
MEN1 O00255 2/20 0.40
LMNA P02545 2/20 0.40
KMT2A Q03164 2/20 0.40
LTB4R Q15722 2/20 0.40
LTB4R2 Q9NPC1 2/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
FBP1 P09467 1/20 0.40
GLA P06280 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29440131 1.00 PDE4A (0.45) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL143031 0.82 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL140388 0.82 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL140387 0.82 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL10611120 0.81 MAPK1 (0.52) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL10611123 0.81 MAPK1 (0.52) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL4273797 0.80 HSD17B2 (0.55) PDE4APDE4BPDE4CPDE4DHTT
SCHEMBL9514114 0.77 HTT (0.54) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL9514123 0.77 HTT (0.54) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL110599 0.76 F2 (0.48) KDM4EHTTRAB9AF2PLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107162928-B Halogenated analogs of anti-fibrotic agents 塞尔塔医疗有限公司 2022-03-11 CN disclosed
EP-3045170-A1 HALOGENATED ANALOGUES OF ANTI-FIBROTIC AGENTS Fibrotech Therapeutics PTY LTD (AU) 2016-07-20 EP disclosed
EP-2220028-B1 HALOGENATED ANALOGUES OF ANTI-FIBROTIC AGENTS FIBROTECH THERAPEUTICS PTY LTD (AU) 2016-03-09 EP disclosed
US-8624056-B2 Halogenated analogues of anti-fibrotic agents FIBROTECH THERAPEUTICS PTY LTD 2014-01-07 US disclosed