SCHEMBL15417831

SCHEMBL15417831

CC(=O)N1CC2CNC(C2)C1

nearest known ligand 0.64

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 19/20 0.64
CHRNA4 P43681 19/20 0.64
CHRNA3 P32297 18/20 0.64
CHRNB4 P30926 17/20 0.64
CHRNA7 P36544 16/20 0.64
CHRNB3 Q05901 1/20 0.59
CHRNA6 Q15825 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1710983 1.00 CHRNB2 (0.64) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA7
SCHEMBL1711288 1.00 CHRNB2 (0.64) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA7
SCHEMBL18828709 0.85 CHRNB2 (0.56) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA7
SCHEMBL3240417 0.83 CHRNB2 (0.52) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA7
SCHEMBL3363292 0.82 CHRNB2 (0.66) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA7
SCHEMBL3333418 0.82 CHRNB2 (0.66) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA7
SCHEMBL31630839 0.82 CHRNB2 (0.66) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA7
SCHEMBL1711422 0.80 CHRNB2 (0.67) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA7
SCHEMBL1711502 0.80 CHRNB2 (0.67) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA7
SCHEMBL14804553 0.80 CHRNB2 (0.58) CHRNB2CHRNA4CHRNA3CHRNB4CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8623857-B2 N-phenyl imidazole carboxamide inhibitors of 3-phosphoinositide-dependent protein kinase-1 MERCK SHARP & DOHME CORP. (US) 2014-01-07 US disclosed