SCHEMBL15418979

SCHEMBL15418979

CC(NC(=O)c1c(O)c2ccc(-c3ccc(Cl)cc3)cc2n(C)c1=O)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 12/20 0.52
L3MBTL1 Q9Y468 1/20 0.50
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
GSK3B P49841 2/20 0.48
EGLN1 Q9GZT9 1/20 0.46
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15419094 0.91 L3MBTL1 (0.57) HIF1AL3MBTL1MEN1KMT2AEGLN1
SCHEMBL15419109 0.91 L3MBTL1 (0.52) HIF1AL3MBTL1MEN1KMT2AEGLN1
SCHEMBL15419125 0.91 HIF1A (0.56) HIF1AL3MBTL1MEN1KMT2AGSK3B
SCHEMBL2382749 0.83 L3MBTL1 (0.55) HIF1AL3MBTL1MEN1KMT2AEGLN1
SCHEMBL2382746 0.83 L3MBTL1 (0.55) HIF1AL3MBTL1MEN1KMT2AEGLN1
SCHEMBL2384965 0.83 L3MBTL1 (0.57) HIF1AL3MBTL1MEN1KMT2A
SCHEMBL2384968 0.83 L3MBTL1 (0.57) HIF1AL3MBTL1MEN1KMT2A
SCHEMBL2382306 0.82 EGLN1 (0.67) HIF1AL3MBTL1MEN1KMT2AGSK3B
SCHEMBL2383427 0.82 L3MBTL1 (0.54) HIF1AL3MBTL1MEN1KMT2AEGLN1
SCHEMBL2382301 0.82 EGLN1 (0.67) HIF1AL3MBTL1MEN1KMT2AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960363-B1 QUINOLONE BASED COMPOUNDS EXHIBITING PROLYL HYDROXYLASE INHIBITORY ACTIVITY, COMPOSITIONS AND USES THEREOF AMGEN INC (US) 2014-01-22 EP claimed