SCHEMBL15423980

SCHEMBL15423980

[2H]c1c(C)c([2H])c(C([2H])[2H])c(N)c1C([2H])[2H]

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
TDP1 Q9NUW8 2/20 0.38
TP53 P04637 1/20 0.38
CYP3A4 P08684 1/20 0.38
TSHR P16473 1/20 0.38
POLB P06746 1/20 0.32
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31620975 0.65 ALDH1A1 (0.60) ALDH1A1TDP1TP53CYP3A4TSHR
SCHEMBL15423981 0.65 ALDH1A1 (0.52) ALDH1A1TDP1TP53CYP3A4TSHR
SCHEMBL15423982 0.64 ALDH1A1 (0.39) ALDH1A1TDP1TP53CYP3A4TSHR
SCHEMBL11791406 0.63
SCHEMBL2296346 0.62 ALDH1A1 (0.36) ALDH1A1TDP1TP53CYP3A4TSHR
SCHEMBL29701329 0.62 ALDH1A1 (0.70) ALDH1A1TDP1TP53CYP3A4TSHR
SCHEMBL139002 0.61 ALDH1A1 (0.65) ALDH1A1TDP1TP53CYP3A4TSHR
SCHEMBL14825817 0.61 CYP3A4 (0.40) ALDH1A1TDP1TP53CYP3A4TSHR
SCHEMBL12024356 0.59 POLB (0.40) ALDH1A1TDP1TP53CYP3A4TSHR
SCHEMBL12559554 0.59

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140018379-A1 PYRIMIDINE DERIVATIVES CONCERT PHARMACEUTICALS INC. (US) 2014-01-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140018379-A1 PYRIMIDINE DERIVATIVES DPYD, TYMS, TYMP ALDH1A1 518/4885TDP1 300/4885TP53 496/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.