SCHEMBL1542544

SCHEMBL1542544

CCCCc1cc(-c2ccc[nH]c2=O)cc(NC(=O)c2ccc(NS(C)(=O)=O)cc2)c1OC

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.57
KDM4E B2RXH2 1/20 0.46
HPGD P15428 4/20 0.41
MAPK10 P53779 1/20 0.41
ALDH1A1 P00352 5/20 0.41
MAPK1 P28482 1/20 0.41
IDO1 P14902 2/20 0.39
CDK9 P50750 1/20 0.39
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
MAPT P10636 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
LMNA P02545 1/20 0.37
ABL1 P00519 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
F10 P00742 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1542369 0.83 CYP3A4 (0.65) CYP3A4HPGDMAPK10ALDH1A1MAPK1
SCHEMBL1542708 0.82 CYP3A4 (0.48) CYP3A4KDM4EHPGDMAPK10ALDH1A1
SCHEMBL1542546 0.80 CYP3A4 (0.54) CYP3A4CNR1CNR2
SCHEMBL2126941 0.76 CYP3A4 (0.53) CYP3A4KDM4EHPGDMAPK10ALDH1A1
SCHEMBL2129460 0.74 CYP3A4 (0.59) CYP3A4HPGDMAPK10ALDH1A1MAPK1
SCHEMBL2129383 0.73 CYP3A4 (0.53) CYP3A4ALDH1A1CDK9MEN1KMT2A
SCHEMBL2127061 0.73 CYP3A4 (0.53) CYP3A4HPGDALDH1A1CDK9MEN1
SCHEMBL1542581 0.72 CYP3A4 (1.00) CYP3A4
SCHEMBL1542597 0.72 CYP3A4 (0.57) CYP3A4KDM4EHPGDALDH1A1MAPK1
SCHEMBL2128420 0.72 CYP3A4 (0.53) CYP3A4KDM4EHPGDALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2307372-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2011-04-13 EP disclosed