SCHEMBL1542546

SCHEMBL1542546

CCCCc1cc(-c2ccc[nH]c2=O)cc(-c2cc(NS(C)(=O)=O)ccc2C(N)=O)c1OC

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.54
IKBKB O14920 4/20 0.37
CHUK O15111 4/20 0.37
BRD4 O60885 2/20 0.36
NR3C1 P04150 1/20 0.36
CNR2 P34972 7/20 0.35
CNR1 P21554 6/20 0.35
FYN P06241 1/20 0.33
TGFBR1 P36897 1/20 0.33
ACVR1 Q04771 1/20 0.33
PDPK1 O15530 1/20 0.33
EP300 Q09472 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1542544 0.80 CYP3A4 (0.57) CYP3A4CNR2CNR1
SCHEMBL1542988 0.71 CYP3A4 (0.81) CYP3A4BRD4PDPK1EP300
SCHEMBL1542581 0.70 CYP3A4 (1.00) CYP3A4BRD4EP300
SCHEMBL1542304 0.70 CYP3A4 (0.79) CYP3A4BRD4PDPK1EP300
SCHEMBL1542623 0.69 CYP3A4 (0.72) CYP3A4PDPK1EP300
SCHEMBL2128400 0.69 CYP3A4 (0.84) CYP3A4IKBKBBRD4NR3C1FYN
SCHEMBL1542682 0.69 CYP3A4 (0.69) CYP3A4IKBKBCHUKEP300
SCHEMBL1542941 0.68 CYP3A4 (0.41) CYP3A4IKBKBCHUKCNR2
SCHEMBL1542813 0.67 CYP3A4 (0.77) CYP3A4BRD4FYNTGFBR1ACVR1
SCHEMBL1542597 0.67 CYP3A4 (0.57) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2307372-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2011-04-13 EP disclosed